SCHEMBL626795

SCHEMBL626795

CC(=O)OC1CCC(Nc2nn3c(Cl)c(-c4cnc(N)c(C(F)(F)F)c4)nc3s2)CC1

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 11/20 0.41
CYP3A4 P08684 1/20 0.41
PIK3CD O00329 2/20 0.38
PIK3CB P42338 2/20 0.38
PIK3CG P48736 2/20 0.38
PIK3C3 Q8NEB9 1/20 0.38
PI4KB Q9UBF8 1/20 0.38
MAP3K12 Q12852 2/20 0.37
FYN P06241 6/20 0.37
HASPIN Q8TF76 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL626796 0.89 PIK3CA (0.39) PIK3CACYP3A4PIK3CDPIK3CBPIK3CG
SCHEMBL627322 0.88 FYN (0.48) PIK3CACYP3A4PIK3CDPIK3CBPIK3CG
SCHEMBL627467 0.87 HASPIN (0.43) PIK3CACYP3A4PIK3CDPIK3CBPIK3CG
SCHEMBL626189 0.84 MAP3K12 (0.42) PIK3CAMAP3K12
SCHEMBL628258 0.81 DPP4 (0.38) PIK3CACYP3A4PIK3CDPIK3CBPIK3CG
SCHEMBL627321 0.76 FYN (0.48) PIK3CACYP3A4PIK3CDPIK3CBPIK3CG
SCHEMBL627323 0.76 FYN (0.48) PIK3CACYP3A4PIK3CDPIK3CBPIK3CG
SCHEMBL627396 0.75 PIK3CA (0.53) PIK3CAFYNHASPIN
SCHEMBL627398 0.75 PIK3CA (0.53) PIK3CAFYNHASPIN
SCHEMBL627466 0.75 HASPIN (0.43) PIK3CACYP3A4PIK3CDPIK3CBPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012020215-A1 AMINO- IMIDAZOLOTHIADIAZOLES FOR USE AS PROTEIN OR LIPID KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLÓGICAS (CNIO) (ES) 2012-02-16 WO disclosed