SCHEMBL6270795

SCHEMBL6270795

C=CCc1nc2nc(N)nc(Cl)c2[nH]1

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 1/20 0.40
CDK1 P06493 3/20 0.34
CCNB1 P14635 3/20 0.34
CCNA2 P20248 3/20 0.34
CDK2 P24941 3/20 0.34
CCNA1 P78396 2/20 0.34
MGMT P16455 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
PNP P00491 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7063134 0.83 PDPK1 (0.37) CDK1CCNB1CCNA2CDK2CCNA1
SCHEMBL1344340 0.77 NPSR1 (0.34) CDK1CCNB1CCNA2CDK2CCNA1
SCHEMBL6533716 0.74 EGLN1 (0.39)
SCHEMBL669005 0.74 PNP (0.59) NPSR1PNP
SCHEMBL2098711 0.74 DPP4 (0.44) DPP4CDK1CCNB1CCNA2CDK2
SCHEMBL6356987 0.71 PNP (0.54) DPP4PNP
SCHEMBL3158628 0.71 DPP4 (0.50) DPP4PNP
SCHEMBL17574491 0.71 NPSR1 (0.36) NPSR1PNP
SCHEMBL1101441 0.70 NPSR1 (0.41) NPSR1
SCHEMBL1101374 0.69 NPSR1 (0.40) NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1017394-B1 CYCLIN DEPENDENT KINASE INHIBITING PURINE DERIVATIVES CANCER REC TECH LTD (GB) 2005-12-07 EP disclosed
US-6303618-B1 ADMINISTERING PURINE COMPOUND WHICH INHIBITS CYCLIC DEPENDENT KINASE ACTIVITY FOR THERAPY OF TUMOR OR OTHER CELL PROLIFERATION DISORDER CANCER RESEARCH CAMPAIGN TECHNOLOGY LIMITED (GB) 2001-10-16 US disclosed
EP-1017394-A1 CYCLIN DEPENDENT KINASE INHIBITING PURINE DERIVATIVES CANCER RESEARCH CAMPAIGN TECHNOLOGY LIMITED (GB) 2000-07-12 EP disclosed
WO-1999002162-A9 CYCLIN DEPENDENT KINASE INHIBITING PURINE DERIVATIVES CANCER RES CAMPAIGN TECH (GB) 1999-07-29 WO disclosed
WO-1999002162-A1 CYCLIN DEPENDENT KINASE INHIBITING PURINE DERIVATIVES CANCER RESEARCH CAMPAIGN TECHNOLOGY LIMITED (GB) 1999-01-21 WO disclosed