SCHEMBL6272901

SCHEMBL6272901

CC(C(=O)O)c1cccc(-c2ccc(OC(F)(F)F)cc2)c1

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 5/20 0.52
PTGS1 P23219 1/20 0.50
F9 P00740 1/20 0.50
AKR1C3 P42330 6/20 0.49
AKR1C2 P52895 6/20 0.49
AKR1C4 P17516 1/20 0.49
AKR1C1 Q04828 1/20 0.49
MMP12 P39900 2/20 0.48
MMP13 P45452 1/20 0.48
RXRA P19793 1/20 0.47
RXRB P28702 1/20 0.47
RXRG P48443 1/20 0.47
APP P05067 1/20 0.46
CYP2C19 P33261 1/20 0.46
AURKA O14965 1/20 0.46
TPX2 Q9ULW0 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1123024 0.86 PTGS2 (0.59) PTGS2PTGS1AKR1C3AKR1C2AKR1C1
SCHEMBL1759907 0.84 PTGS1 (0.65) PTGS2PTGS1AKR1C3AKR1C2AKR1C4
SCHEMBL29537690 0.84 PTGS1 (0.65) PTGS2PTGS1AKR1C3AKR1C2AKR1C4
SCHEMBL1991313 0.84 PTGS1 (0.65) PTGS2PTGS1AKR1C3AKR1C2AKR1C4
SCHEMBL18069753 0.84 F9 (0.48) F9AKR1C2AKR1C1MMP12MMP13
SCHEMBL22888490 0.83 PTPN5 (0.54) F9MMP12MMP13RXRARXRB
SCHEMBL14603498 0.82 F9 (0.47) F9AKR1C2AKR1C1MMP12MMP13
SCHEMBL6270587 0.82 AKR1C3 (0.63) PTGS2AKR1C3AKR1C2AKR1C4AKR1C1
SCHEMBL9680427 0.81 PTGS2 (0.50) PTGS2PTGS1AKR1C3AKR1C2APP
SCHEMBL9680432 0.81 PTGS2 (0.50) PTGS2PTGS1AKR1C3AKR1C2APP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1604970-A1 2-(Biphenyl-3-yl)-carboxylic acids of gamma-secretase-modulating activity CELLZOME AG (DE) 2005-12-14 EP disclosed
WO-2005110963-A1 (BIPHENYL-3-YL)-CARBOXYLIC ACIDS AND DERIVATIVES THEREOF AND THEIR USE IN THERAPY CELLZOME AG (DE) 2005-11-24 WO disclosed