SCHEMBL6273563

SCHEMBL6273563

Oc1ccc(-c2[nH]nc(C(F)(F)F)c2-c2ccc(Cl)cc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RPS6KA3 P51812 3/20 0.46
PLK4 O00444 2/20 0.46
DAPK3 O43293 2/20 0.46
DYRK3 O43781 2/20 0.46
ROCK2 O75116 2/20 0.46
PRKD3 O94806 2/20 0.46
MAP4K4 O95819 2/20 0.46
RET P07949 2/20 0.46
FER P16591 2/20 0.46
RPS6KB1 P23443 2/20 0.46
CDK2 P24941 2/20 0.46
MARK3 P27448 2/20 0.46
GSK3B P49841 2/20 0.46
LIMK1 P53667 2/20 0.46
MAP4K2 Q12851 2/20 0.46
STK3 Q13188 2/20 0.46
ROCK1 Q13464 2/20 0.46
CAMK2B Q13554 2/20 0.46
CAMK2G Q13555 2/20 0.46
CAMK2D Q13557 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16797093 0.82 NPSR1 (0.46) DYRK1AMAPK1FLT3MEN1MAPT
SCHEMBL8593143 0.75 NPSR1 (0.43) GSK3BCDK1CDK5GYS1MEN1
SCHEMBL1279682 0.75 IKBKB (0.46) MKNK2MAPK1GYS1MEN1MAPT
SCHEMBL28724776 0.72 GRM5 (0.44) MAPK1MEN1MAPTHTTKMT2A
SCHEMBL14519434 0.72 MAPK14 (0.64) PRKD3MAP4K4GSK3BPRKD2CLK4
SCHEMBL30639562 0.70 MAPT (0.46) RPS6KA3PLK4DAPK3DYRK3ROCK2
SCHEMBL2698649 0.70 MAPK1 (0.44) RPS6KA3PLK4DAPK3DYRK3ROCK2
SCHEMBL8195709 0.69 GSK3B (0.41) RPS6KA3PLK4DAPK3DYRK3ROCK2
SCHEMBL6180483 0.68 PTGS2 (0.53) CSNK1DMAPK11MAPK14SMN1; SMN2
SCHEMBL8764358 0.68 PTGS2 (0.52) MAPK1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005037227-A2 SELECTIVE COX-2 INHIBITORS MICROBIA, INC. (US) 2005-04-28 WO claimed