SCHEMBL6273576

SCHEMBL6273576

O=C(NCCO)c1cc(S(=O)(=O)c2ccc(CCN(Cc3ccccc3)C[C@@H](O)c3ccc(Cl)nc3)cc2)ccc1OCc1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 2/20 0.37
LRRK2 Q5S007 2/20 0.37
POLB P06746 1/20 0.37
KMT2A Q03164 1/20 0.36
GLP1R P43220 1/20 0.35
GCGR P47871 1/20 0.35
LMNA P02545 1/20 0.35
PKM P14618 1/20 0.35
SLC12A2 P55011 1/20 0.35
SLC12A5 Q9H2X9 1/20 0.35
TRPM8 Q7Z2W7 1/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
CYP2C9 P11712 2/20 0.35
NAMPT P43490 1/20 0.35
KCNH2 Q12809 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C19 P33261 1/20 0.34
CCR2 P41597 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6273580 1.00 AKR1C3 (0.37) AKR1C3LRRK2POLBKMT2AGLP1R
SCHEMBL6269051 0.92 LRRK2 (0.39) AKR1C3LRRK2POLBKMT2ALMNA
SCHEMBL6269043 0.92 LRRK2 (0.39) AKR1C3LRRK2POLBKMT2ALMNA
SCHEMBL6269814 0.92 LRRK2 (0.40) AKR1C3LRRK2POLBLMNAPKM
SCHEMBL6269808 0.92 LRRK2 (0.40) AKR1C3LRRK2POLBLMNAPKM
SCHEMBL6272707 0.91 LRRK2 (0.40) AKR1C3LRRK2KMT2ACYP2C9NAMPT
SCHEMBL6272709 0.91 LRRK2 (0.40) AKR1C3LRRK2KMT2ACYP2C9NAMPT
SCHEMBL6267521 0.90 AKR1C3 (0.40) AKR1C3LRRK2POLBKMT2ASPHK2
SCHEMBL6267524 0.90 AKR1C3 (0.40) AKR1C3LRRK2POLBKMT2ASPHK2
SCHEMBL6272461 0.89 PTPN2 (0.40) LRRK2KMT2ALMNASMN1; SMN2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005110981-A1 AMINOALCOHOL DERIVATIVES ASTELLAS PHARMA INC. (JP) 2005-11-24 WO disclosed