SCHEMBL6274969

SCHEMBL6274969

Oc1cncc2c1cnn2-c1cccc(F)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.45
CYP17A1 P05093 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP11B2 P19099 4/20 0.43
MAPK14 Q16539 3/20 0.42
CCR1 P32246 3/20 0.42
CYP11B1 P15538 2/20 0.41
GSK3B P49841 1/20 0.39
SLC2A1 P11166 1/20 0.39
SLC2A2 P11168 1/20 0.39
SLC2A3 P11169 1/20 0.39
NPC1 O15118 2/20 0.39
SMO Q99835 1/20 0.38
NR3C1 P04150 2/20 0.38
PGR P06401 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
KDM4E B2RXH2 1/20 0.38
MAPT P10636 1/20 0.38
RAB9A P51151 1/20 0.38
CYP3A4 P08684 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6278822 0.83 RXFP1 (0.45) ESR1CYP17A1CYP1A2CYP11B2MAPK14
SCHEMBL6267646 0.83 NPC1 (0.48) CYP11B2CYP11B1NPC1KDM4EMAPT
SCHEMBL31632994 0.74 CYP11B2 (0.48) ESR1CYP11B2MAPK14CYP11B1NPC1
SCHEMBL4573821 0.74 MAPK14 (0.50) ESR1CYP17A1CYP1A2CYP11B2MAPK14
SCHEMBL31632913 0.72 CCR1 (0.58) CYP17A1CYP1A2CYP11B2MAPK14CCR1
SCHEMBL2207105 0.72 CCR1 (0.58) CYP11B2CCR1CYP3A4
SCHEMBL30918020 0.71 CYP11B2 (0.54) CYP11B2MAPK14CYP11B1SMONR3C1
SCHEMBL31632873 0.70 CCR1 (0.46) CYP17A1CYP1A2CYP11B2MAPK14CCR1
SCHEMBL6207703 0.70 SLC2A1 (0.58) CYP17A1CYP1A2GSK3BSLC2A1SLC2A2
SCHEMBL31632924 0.70 MAPK14 (0.50) MAPK14CCR1SLC2A1SLC2A2SLC2A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1551841-A1 PYRAZOLOPYRIMIDINES AS KINASE INHIBITORS SmithKline Beecham Corporation (US) 2005-07-13 EP disclosed
WO-2004009602-A1 PYRAZOLOPYRIMIDINES AS KINASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2004-01-29 WO disclosed