SCHEMBL6280385

SCHEMBL6280385

COc1cc(N[C@@H](C)CCCNC(=O)C(C)N)c2nc(C(C)(C)C)ccc2c1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 2/20 0.48
HSP90AB1 P08238 2/20 0.48
KDM4E B2RXH2 3/20 0.47
CASP1 P29466 2/20 0.47
THRB P10828 2/20 0.47
RAD52 P43351 1/20 0.47
CASP7 P55210 1/20 0.47
CASP6 P55212 1/20 0.47
CASP8 Q14790 1/20 0.47
CYP1A2 P05177 2/20 0.47
ALDH1A1 P00352 2/20 0.47
ABCB11 O95342 1/20 0.47
ESR1 P03372 1/20 0.47
PGR P06401 1/20 0.47
ADRB2 P07550 1/20 0.47
CHRM2 P08172 1/20 0.47
ADRB1 P08588 1/20 0.47
HTR1A P08908 1/20 0.47
ADRA2A P08913 1/20 0.47
ADORA3 P0DMS8 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6280393 1.00 HSP90AA1 (0.48) HSP90AA1HSP90AB1KDM4ECASP1THRB
SCHEMBL4727368 1.00 HSP90AA1 (0.48) HSP90AA1HSP90AB1KDM4ECASP1THRB
SCHEMBL5086470 0.93 HSP90AA1 (0.46) HSP90AA1HSP90AB1KDM4ECASP1THRB
SCHEMBL5086556 0.90 KDM4E (0.52) HSP90AA1HSP90AB1KDM4ECASP1THRB
SCHEMBL4729756 0.90 KDM4E (0.49) HSP90AA1HSP90AB1KDM4ECASP1THRB
SCHEMBL4727369 0.85 KDM4E (0.48) HSP90AA1HSP90AB1KDM4ECASP1THRB
SCHEMBL5086463 0.84 HSP90AA1 (0.51) HSP90AA1HSP90AB1KDM4ECASP1THRB
SCHEMBL6268435 0.83 KDM4E (0.47) HSP90AA1HSP90AB1KDM4ECASP1THRB
SCHEMBL5080647 0.83 MAOA (0.66) HSP90AA1HSP90AB1KDM4ECASP1THRB
SCHEMBL6276764 0.82 KDM4E (0.46) HSP90AA1HSP90AB1KDM4ECASP1THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1606263-A1 RING-SUBSTITUTED 8-AMINOQUINOLINE DERIVATIVES AS ANTIMALARIAL AGENTS Council of Scientific and Industrial Research (IN) 2005-12-21 EP disclosed
WO-2004085402-A1 RING-SUBSTITUTED 8-AMINOQUNOLINE DERIVATES AS ANTIMALARIAL AGENTS COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2004-10-07 WO disclosed