SCHEMBL6286665

SCHEMBL6286665

N#C/C(=C\c1ccc(O)c(O)c1)C(=O)O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 11/20 1.00
KDM4E B2RXH2 9/20 0.73
ALDH1A1 P00352 8/20 0.73
HPGD P15428 7/20 0.73
MEN1 O00255 7/20 0.73
KMT2A Q03164 7/20 0.73
ERBB2 P04626 6/20 0.73
MAPT P10636 6/20 0.73
TDP1 Q9NUW8 6/20 0.73
TP53 P04637 5/20 0.73
HSD17B10 Q99714 5/20 0.73
CYP1A2 P05177 4/20 0.73
LCK P06239 1/20 0.73
CYP3A4 P08684 5/20 0.69
BLM P54132 5/20 0.69
ALOX15 P16050 4/20 0.69
ALOX12 P18054 4/20 0.69
MAPK1 P28482 4/20 0.69
PMP22 Q01453 4/20 0.69
RECQL P46063 4/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29483469 1.00 EGFR (1.00) EGFRKDM4EALDH1A1HPGDMEN1
SCHEMBL29357482 1.00 EGFR (1.00) EGFRKDM4EALDH1A1HPGDMEN1
SCHEMBL5908882 1.00 EGFR (1.00) EGFRKDM4EALDH1A1HPGDMEN1
SCHEMBL17457139 1.00 EGFR (1.00) EGFRKDM4EALDH1A1HPGDMEN1
SCHEMBL13060220 0.87 EGFR (0.77) EGFRKDM4EALDH1A1HPGDMEN1
SCHEMBL20995953 0.85 EGFR (0.74) EGFRKDM4EALDH1A1HPGDMEN1
SCHEMBL20995956 0.85 EGFR (0.74) EGFRKDM4EALDH1A1HPGDMEN1
SCHEMBL10241964 0.85 EGFR (0.74) EGFRKDM4EALDH1A1HPGDMEN1
SCHEMBL1705642 0.85 EGFR (1.00) EGFRKDM4EALDH1A1HPGDMEN1
SCHEMBL6285299 0.85 EGFR (1.00) EGFRKDM4EALDH1A1HPGDMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 36 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2235852-A None JP disclosed
EP-4739310-A1 ECTONUCLEOTIDE PYROPHOSPHATASE/PHOSPHODIESTERASE 1 (ENPP1) INHIBITOR COMBINATIONS AND USES THEREOF Insilico Medicine IP Limited (HK) 2026-05-13 EP disclosed
EP-4578457-A1 PHARMACEUTICAL FOR TREATING AND/OR PREVENTING CANCER Toray Industries, Inc. (JP) 2025-07-02 EP disclosed
CN-119768182-A Medicine for treating and/or preventing cancer 东丽株式会社 2025-04-04 CN disclosed
WO-2025051110-A1 COMBINATIONS TREATMENTS OF DIACYLGLYCEROL KINASE (DGK) ALPHA INHIBITORS AND OTHER THERAPIES INSILICO MEDICINE IP LIMITED (CN) 2025-03-13 WO disclosed
WO-2025007955-A1 ECTONUCLEOTIDE PYROPHOSPHATASE/PHOSPHODIESTERASE 1 (ENPP1) INHIBITOR COMBINATIONS AND USES THEREOF INSILICO MEDICINE IP LIMITED (CN) 2025-01-09 WO disclosed
WO-2024217502-A1 METHIONINE ADENOSYLTRANSFERASE 2A (MAT2A) INHIBITOR COMBINATIONS AND USES THEREOF INSILICO MEDICINE IP LIMITED (CN) 2024-10-24 WO disclosed
WO-2024178274-A2 METHODS OF DEGRADING RAF(RAF) PROTEIN IN CELLS USING MITOGEN-ACTIVATED PROTEIN KINASE KINASE 1/2 (MEK1/2) PROTEIN DEGRADERS INSTITUTE FOR CANCER RESEARCH D/B/A THE RESEARCH INSTITUTE OF FOX CHASE CANCER CENTER (US) 2024-08-29 WO disclosed
CN-114656372-B P-phenylenediamine bridging compound and application thereof in preparation of medicines for treating sugar metabolism disorder diseases 广州药本君安医药科技股份有限公司 2024-06-18 CN disclosed
CN-114573476-B Linear head-tail diamine bridging compound and application thereof in preparation of medicines for treating sugar metabolic disorder diseases 广州药本君安医药科技股份有限公司 2024-06-11 CN disclosed
EP-0322738-B1 Benzylidene-malononitrile derivatives for the inhibition of proliferative processes in mammalian cells YISSUM RES DEV CO (IL) 1995-04-12 EP disclosed
EP-0614661-A2 Benzylidene- and cinnamylidine-malononitrile derivatives for the inhibition of proliferative processes in mammalian cells YISSUM RESEARCH DEVELOPMENT COMPANY OF THE HEBREW UNIVERSITY OF JERUSALEM (IL) 1994-09-14 EP disclosed
EP-0339671-B1 Derivative of caffeic acid and pharmaceutical composition containing the same SUNTORY LTD (JP) 1994-08-10 EP disclosed
EP-0572167-A1 Cosmestic composition UNILEVER PLC (GB) 1993-12-01 EP disclosed
US-5217999-A Antigrowth agents YISSUM RESEARCH DEVELOPMENT COMPANY OF THE HEBREW UNIVERSITY OF JERUSALEM (IL) 1993-06-08 US disclosed
WO-1991016892-A1 STYRYL COMPOUNDS WHICH INHIBIT EGF RECEPTOR PROTEIN TYROSINE KINASE RORER INTERNATIONAL (HOLDINGS), INC. (US) 1991-11-14 WO disclosed
US-5063243-A Arteriosclerosis treatment SUNTORY, LTD. (JP) 1991-11-05 US disclosed
JP-H02235852-A CAFFEIC ACID DERIVATIVE AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME SUNTORY LTD 1990-09-18 JP disclosed
EP-0339671-A2 Derivative of caffeic acid and pharmaceutical composition containing the same SUNTORY LIMITED (JP) 1989-11-02 EP disclosed
EP-0322738-A2 Benzylidene-malononitrile derivatives for the inhibition of proliferative processes in mammalian cells YISSUM RESEARCH DEVELOPMENT COMPANY OF THE HEBREW UNIVERSITY OF JERUSALEM (IL) 1989-07-05 EP disclosed