SCHEMBL6288762

SCHEMBL6288762

c1ccc(P(c2ccccc2)c2nc(P(c3ccccc3)c3ccccc3)nc(P(c3ccccc3)c3ccccc3)n2)cc1

nearest known ligand 0.61

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.61
TDP1 Q9NUW8 1/20 0.61
KDM4E B2RXH2 1/20 0.46
GAA P10253 1/20 0.46
ESR1 P03372 4/20 0.46
ESR2 Q92731 4/20 0.46
NPSR1 Q6W5P4 1/20 0.36
MAPT P10636 1/20 0.33
MEN1 O00255 1/20 0.32
RAB9A P51151 1/20 0.32
KMT2A Q03164 1/20 0.32
CYP2A6 P11509 1/20 0.32
ALOX12 P18054 1/20 0.32
DRD1 P21728 2/20 0.31
ALDH1A1 P00352 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9332945 0.88 TDP1 (0.48) CYP3A4TDP1KDM4EGAAESR1
SCHEMBL9335851 0.85 CYP3A4 (0.50) CYP3A4TDP1KDM4EGAAESR1
SCHEMBL9336100 0.83 CYP3A4 (0.48) CYP3A4TDP1KDM4EGAAESR1
SCHEMBL14735869 0.81 TDP1 (0.92) CYP3A4TDP1KDM4EGAAESR1
SCHEMBL10819825 0.78 KDM4E (0.60) CYP3A4TDP1KDM4EGAAESR1
SCHEMBL2085135 0.77 TDP1 (1.00) CYP3A4TDP1KDM4EGAAESR1
Benzene SCHEMBL6890099 0.77 TDP1 (1.00) CYP3A4TDP1KDM4EGAAESR1
SCHEMBL5028587 0.77 TDP1 (1.00) CYP3A4TDP1KDM4EGAAESR1
SCHEMBL101 0.77 TDP1 (1.00) CYP3A4TDP1KDM4EGAAESR1
SCHEMBL25384985 0.74 TDP1 (0.92) CYP3A4TDP1KDM4EGAAESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20020137820-A1 Phosphorus compounds SANDOZ LTD. (CH) 2002-09-26 US claimed
US-6864304-B2 Phosphorus compounds CLARIANT FINANCE (BVI) LIMITED (VG) 2005-03-08 US disclosed
US-20020137820-A1 Phosphorus compounds SANDOZ LTD. (CH) 2002-09-26 US disclosed
US-6369140-B1 POLYOLEFIN AND PHOSPHINE OR PHOSPHORANE COMPOUNDS STABILIZERS; OXIDATION, HEAT, STRESS, AND ULTRAVIOLET RADIATION RESISTANCE CLARIANT FINANCE (BVI) LIMITED (BV) 2002-04-09 US disclosed
US-5488079-A HEAT AND LIGHT STABILIZERS FOR OLEFINS USING PHOSPHINES SANDOZ LTD. (CH) 1996-01-30 US disclosed
EP-0499329-B1 Carbonylation catalyst system SHELL INT RESEARCH (NL) 1994-05-04 EP disclosed
US-5258546-A Reaction of acetylene with carbon monoxide for alpha, beta-olefin unsaturated compounds SHELL OIL COMPANY (US) 1993-11-02 US disclosed
US-5189003-A Of group 8 metal or compound and a polyphosphine SHELL OIL COMPANY (US) 1993-02-23 US disclosed
EP-0499329-A1 Carbonylation catalyst system SHELL INTERNATIONALE RESEARCHMAATSCHAPPIJ B.V. (NL) 1992-08-19 EP disclosed