SCHEMBL6289101

SCHEMBL6289101

COC(=O)c1ccc(CNC(=O)CCCC(=O)NCCCN(C)CCNC(=O)CCCC(=O)NCc2ccc(C(=O)OC)c(O)c2)cc1O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 11/20 0.49
EGFR P00533 1/20 0.48
SRC P12931 1/20 0.48
CYP1A2 P05177 4/20 0.43
CYP3A4 P08684 4/20 0.43
ALDH1A1 P00352 3/20 0.43
CYP2D6 P10635 3/20 0.43
CYP2C9 P11712 3/20 0.43
CYP2C19 P33261 3/20 0.43
ALOX15 P16050 2/20 0.43
BLM P54132 2/20 0.43
PMP22 Q01453 2/20 0.43
HPGD P15428 1/20 0.43
APP P05067 1/20 0.42
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
KDM1A O60341 1/20 0.41
NR1I2 O75469 1/20 0.41
LMNA P02545 1/20 0.41
ALOX5 P09917 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6289048 0.82 TRPV1 (0.57) TRPV1EGFRSRCCYP1A2CYP3A4
SCHEMBL6290018 0.77 CA1 (0.42) TRPV1EGFRSRCCYP1A2CYP3A4
SCHEMBL6290007 0.74 CA1 (0.41) TRPV1EGFRSRCMEN1KMT2A
SCHEMBL7731012 0.72 EGFR (0.39) TRPV1EGFRSRCCYP1A2CYP3A4
SCHEMBL14401631 0.72 SMN1; SMN2 (0.56) TRPV1EGFRSRCALDH1A1BLM
Hydrochloric Acid SCHEMBL6292854 0.69 CA12 (0.59) TRPV1EGFRSRCALDH1A1ALOX15
SCHEMBL6289111 0.69 EGFR (0.41) TRPV1EGFRSRCCYP1A2CYP3A4
SCHEMBL6290003 0.69 EGFR (0.51) TRPV1EGFRSRCCYP1A2CYP3A4
SCHEMBL13024608 0.68 CA12 (0.50) TRPV1EGFRSRCALDH1A1ALOX15
SCHEMBL12857040 0.68 CA12 (0.61) EGFRSRCCYP3A4ALDH1A1ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6870065-B2 Bifunctional boronic compound complexing reagents and complexes CAMBREX BIO SCIENCE ROCKLAND, INC. (US) 2005-03-22 US disclosed
US-6414122-B1 BIOCHEMICAL CONJUGATION TO PROTEINS, PEPTIDES, HORMONES, POLYSACCHARIDES, NUCLEIC ACIDS, LIPOSOMES, RADIONUCLIDES, HAPTENS, AND TOXINS PROLINX, INC. 2002-07-02 US disclosed
US-6156884-A Bifunctional boronic compound complexing reagents and complexes PROLINX, INC. (US) 2000-12-05 US disclosed