SCHEMBL7731012

SCHEMBL7731012

COC(=O)c1ccc(CCNC(=O)CCCC(=O)NCCN(CCNC(=O)CCCC(=O)NCc2ccc(C(=O)OC)c(O)c2)C(=O)CCCC(=O)NN(C=O)OC(C)(C)C)cc1O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.39
SRC P12931 1/20 0.39
TRPV1 Q8NER1 8/20 0.37
MAPT P10636 4/20 0.36
HSD17B10 Q99714 2/20 0.36
CNR1 P21554 2/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
HPGD P15428 2/20 0.35
KDM4E B2RXH2 1/20 0.35
NPC1 O15118 1/20 0.35
GMNN O75496 1/20 0.35
USP2 O75604 1/20 0.35
LMNA P02545 1/20 0.35
TP53 P04637 1/20 0.35
CYP1A2 P05177 1/20 0.35
POLB P06746 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
IDE P14735 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6290007 0.83 CA1 (0.41) EGFRSRCTRPV1MAPTHSD17B10
SCHEMBL6290018 0.80 CA1 (0.42) EGFRSRCTRPV1MAPTHSD17B10
SCHEMBL6289101 0.72 TRPV1 (0.49) EGFRSRCTRPV1MAPTHSD17B10
SCHEMBL6290160 0.72 CA1 (0.42) TRPV1CNR1HPGDCYP1A2CYP3A4
SCHEMBL6289111 0.70 EGFR (0.41) EGFRSRCTRPV1MAPTHSD17B10
SCHEMBL6289048 0.69 TRPV1 (0.57) EGFRSRCTRPV1MAPTHSD17B10
SCHEMBL8003356 0.66 CA2 (0.48) EGFRSRCMAPTHSD17B10MEN1
SCHEMBL5200513 0.64 CA1 (0.47) MEN1KMT2A
SCHEMBL6289047 0.62 TRPV1 (0.35) TRPV1CNR1HPGDCYP1A2CYP3A4
SCHEMBL6293459 0.62 CA1 (0.40) TRPV1HPGDCYP1A2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6414122-B1 BIOCHEMICAL CONJUGATION TO PROTEINS, PEPTIDES, HORMONES, POLYSACCHARIDES, NUCLEIC ACIDS, LIPOSOMES, RADIONUCLIDES, HAPTENS, AND TOXINS PROLINX, INC. 2002-07-02 US disclosed
US-6156884-A Bifunctional boronic compound complexing reagents and complexes PROLINX, INC. (US) 2000-12-05 US disclosed