SCHEMBL6294145

SCHEMBL6294145

CCn1ncnc1COc1nn2c(-c3c(F)cccc3F)nnc(C)c2c1C(C)(C)C

nearest known ligand 0.56

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GABRG2 P18507 20/20 0.56
GABRB3 P28472 20/20 0.56
GABRA3 P34903 20/20 0.56
GABRA1 P14867 6/20 0.56
GABRA5 P31644 4/20 0.56
GABRA2 P47869 3/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6293000 0.85 GABRG2 (0.58) GABRG2GABRB3GABRA3GABRA1GABRA5
SCHEMBL2652749 0.81 GABRG2 (0.82) GABRG2GABRB3GABRA3GABRA1GABRA5
SCHEMBL6292561 0.80 GABRG2 (0.56) GABRG2GABRB3GABRA3GABRA1GABRA5
SCHEMBL5230753 0.76 GABRG2 (0.58) GABRG2GABRB3GABRA3GABRA1GABRA5
SCHEMBL5230593 0.75 GABRG2 (0.66) GABRG2GABRB3GABRA3GABRA1GABRA5
SCHEMBL6294094 0.73 GABRG2 (0.70) GABRG2GABRB3GABRA3GABRA1GABRA5
SCHEMBL2655126 0.73 GABRG2 (0.75) GABRG2GABRB3GABRA3GABRA1GABRA5
SCHEMBL2655013 0.73 GABRG2 (0.80) GABRG2GABRB3GABRA3GABRA1
SCHEMBL6292919 0.73 GABRG2 (0.57) GABRG2GABRB3GABRA3GABRA1GABRA5
SCHEMBL2659079 0.73 GABRG2 (0.58) GABRG2GABRB3GABRA3GABRA1GABRA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6872720-B2 Pyrazolo-triazine derivatives as ligands for gaba receptors MERCK SHARP & DOHME LTD. 2005-03-29 US disclosed