SCHEMBL6300639

SCHEMBL6300639

CC(C)(C)[Si](C)(C)OCc1cccc(CNc2ccccn2)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FABP1 P07148 1/20 0.52
FABP6 P51161 1/20 0.52
CXCR4 P61073 1/20 0.50
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
GAA P10253 1/20 0.45
TP53 P04637 1/20 0.45
TSHR P16473 1/20 0.45
KDM4E B2RXH2 1/20 0.45
HIF1A Q16665 1/20 0.44
EPAS1 Q99814 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.43
NOS2 P35228 1/20 0.41
NOS1 P29475 1/20 0.41
NPSR1 Q6W5P4 1/20 0.40
HDAC1 Q13547 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
ALDH1A1 P00352 2/20 0.39
HPGD P15428 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10054969 0.81 FABP1 (0.79) FABP1FABP6CXCR4NPC1RAB9A
SCHEMBL23094637 0.74 MEN1 (0.38) FABP1FABP6CXCR4MEN1KMT2A
SCHEMBL4035843 0.74 CYP2C19 (0.50) FABP1FABP6CXCR4NPC1RAB9A
SCHEMBL6301782 0.74 FABP1 (0.67) FABP1FABP6CXCR4NPC1RAB9A
SCHEMBL6564767 0.74 FABP1 (0.67) FABP1FABP6CXCR4NPC1RAB9A
SCHEMBL11573094 0.74 FABP1 (0.67) FABP1FABP6CXCR4NPC1RAB9A
SCHEMBL11942311 0.73 IDO1 (0.38) TP53
SCHEMBL19892519 0.73 L3MBTL1 (0.61) FABP1FABP6CXCR4NPC1RAB9A
Hydrochloric Acid SCHEMBL6302644 0.73 FABP1 (0.65) FABP1FABP6CXCR4NPC1RAB9A
SCHEMBL15687564 0.72 IDO1 (0.36) TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6846833-B2 Vitronectin receptor antagonist bicyclic compounds, preparation method and compositions containing same LES LABORATORIES SERVIER (FR) 2005-01-25 US disclosed
EP-1268429-B1 VITRONECTIN RECEPTOR ANTAGONIST BICYCLIC COMPOUNDS, PREPARATION METHOD AND COMPOSITIONS CONTAINING SAME SERVIER LAB (FR) 2004-08-18 EP disclosed
EP-1268429-A1 VITRONECTIN RECEPTOR ANTAGONIST BICYCLIC COMPOUNDS, PREPARATION METHOD AND COMPOSITIONS CONTAINING SAME Les Laboratoires Servier (FR) 2003-01-02 EP disclosed
WO-2001079172-A1 VITRONECTIN RECEPTOR ANTAGONIST BICYCLIC COMPOUNDS, PREPARATION METHOD AND COMPOSITIONS CONTAINING SAME LES LABORATOIRES SERVIER Departament Brevets/Fontanes (FR) 2001-10-25 WO disclosed