SCHEMBL6306015

SCHEMBL6306015

CC1Oc2ccc(CN(Cc3cccc(C[N+](C)(C(=O)OC(C)(C)C)c4ccc5c(c4)NC(=O)C(C)O5)c3)C(=O)OC(C)(C)C)cc2NC1=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 8/20 0.42
HSD17B10 Q99714 3/20 0.34
ALOX15 P16050 2/20 0.34
SMYD3 Q9H7B4 2/20 0.33
MAPK1 P28482 2/20 0.32
HDAC3 O15379 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC2 Q92769 1/20 0.32
NCOR2 Q9Y618 1/20 0.32
ALDH1A1 P00352 1/20 0.32
THRB P10828 1/20 0.31
PDE3B Q13370 1/20 0.31
PDE3A Q14432 1/20 0.31
HTR1A P08908 1/20 0.31
HTR7 P34969 1/20 0.31
USP2 O75604 1/20 0.31
GAA P10253 1/20 0.31
KDR P35968 1/20 0.30
HTT P42858 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6304845 0.94 PARP1 (0.39) PARP1HSD17B10ALOX15SMYD3MAPK1
SCHEMBL6302669 0.91 PARP1 (0.32) PARP1HDAC3HDAC1HDAC2NCOR2
SCHEMBL6302932 0.91 PARP1 (0.34) PARP1HSD17B10ALOX15SMYD3
SCHEMBL6303037 0.90 PARP1 (0.36) PARP1HSD17B10ALOX15SMYD3PDE3B
SCHEMBL6305893 0.86 PARP1 (0.54) PARP1HSD17B10ALOX15SMYD3MAPK1
SCHEMBL6309334 0.85 HDAC3 (0.31) HDAC3HDAC1HDAC2NCOR2
SCHEMBL6302634 0.85 PARP1 (0.33) PARP1SMYD3
SCHEMBL7713376 0.84 PARP1 (0.56) PARP1HSD17B10ALOX15SMYD3MAPK1
SCHEMBL6302723 0.83 PARP1 (0.47) PARP1HSD17B10ALOX15SMYD3MAPK1
SCHEMBL6308969 0.82 PARP1 (0.46) PARP1HSD17B10ALOX15SMYD3MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6841550-B1 Benzoxazine and benzothiazine derivatives and their use in medicines SCHERING AKTIENGESELLSCHAFT (DE) 2005-01-11 US disclosed
EP-1114037-B1 BENZOXAZINE AND BENZOTHIAZINE DERIVATIVES AND THEIR USE IN MEDICINES SCHERING AG (DE) 2004-05-12 EP disclosed