SCHEMBL6307449

SCHEMBL6307449

CC(Oc1ccc(O)cc1)C1CCCCN1.O=C(c1c(-c2ccc(O)cc2)noc1-c1ccc(O)cc1)c1c(-c2ccc(O)cc2)noc1-c1ccc(O)cc1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.35
TP53 P04637 1/20 0.33
SLC6A3 Q01959 3/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
DHFR P00374 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
CYP2D6 P10635 1/20 0.33
MAPK1 P28482 1/20 0.33
CYP2C19 P33261 1/20 0.33
HSD17B10 Q99714 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5729286 0.96 PTGS1 (0.34) PTGS1TP53SLC6A3SLC6A2SLC6A4
SCHEMBL5731066 0.94 PTGS1 (0.34) PTGS1TP53ALDH1A1
SCHEMBL5729633 0.93 SLC6A2 (0.37) PTGS1SLC6A3SLC6A2SLC6A4ALDH1A1
SCHEMBL5729513 0.93 SLC6A2 (0.37) PTGS1SLC6A3SLC6A2SLC6A4ALDH1A1
SCHEMBL5729312 0.90 PTGS1 (0.34) PTGS1SLC6A3SLC6A2SLC6A4
SCHEMBL6304492 0.89 MLLT1 (0.34) PTGS1ALDH1A1HPGDCYP2D6MAPK1
SCHEMBL5729044 0.89 SLC6A2 (0.39) PTGS1SLC6A3SLC6A2SLC6A4ALDH1A1
SCHEMBL6307246 0.88 S1PR1 (0.34) SLC6A3SLC6A2SLC6A4
SCHEMBL5729587 0.88 ALDH1A1 (0.38) PTGS1SLC6A3SLC6A2SLC6A4ALDH1A1
SCHEMBL5729015 0.88 ADORA2A (0.33) TP53SLC6A3SLC6A2SLC6A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6869969-B2 Estrogen receptor modulators CHIRON CORPORATION (US) 2005-03-22 US disclosed