SCHEMBL6311149

SCHEMBL6311149

C=C(C(=O)NCCCN1CC(CO)CC1=O)c1ccc(Sc2ccccc2Br)c(Cl)c1

nearest known ligand 0.40

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ITGB2 P05107 16/20 0.40
ICAM1 P05362 16/20 0.40
ITGAL P20701 16/20 0.40
PDE7A Q13946 1/20 0.33
KMT2A Q03164 2/20 0.31
CYP2D6 P10635 1/20 0.31
SMAD3 P84022 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6489137 0.90 ITGB2 (0.41) ITGB2ICAM1ITGALPDE7AKMT2A
SCHEMBL6198619 0.84 ITGB2 (0.57) ITGB2ICAM1ITGALKMT2A
SCHEMBL5830251 0.74 ITGB2 (0.68) ITGB2ICAM1ITGALKMT2A
SCHEMBL5830523 0.72 ITGB2 (0.65) ITGB2ICAM1ITGALKMT2A
SCHEMBL5829934 0.71 EPHX2 (0.40) PDE7AKMT2A
SCHEMBL6196672 0.70 ITGB2 (0.45) ITGB2ICAM1ITGAL
SCHEMBL5830364 0.69 PDE7A (0.38) PDE7AKMT2A
SCHEMBL5829927 0.67 ITGB2 (0.68) ITGB2ICAM1ITGALKMT2A
SCHEMBL6494066 0.67 AKR1C3 (0.40) PDE7AKMT2A
SCHEMBL5830329 0.67 ITGB2 (0.70) ITGB2ICAM1ITGALKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6878700-B1 Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds ABBOTT LABORATORIES (US) 2005-04-12 US disclosed
US-6867203-B2 Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds ABBOTT LABORATORIES (US) 2005-03-15 US disclosed
US-20040116518-A1 Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds ABBOTT LABORATORIES 2004-06-17 US disclosed