SCHEMBL6313858

SCHEMBL6313858

CN(C)c1ccc(C=Cc2nc3ccc(Cl)cc3c(=O)n2Cc2cccc(CN)c2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.51
MEN1 O00255 1/20 0.51
ALDH1A1 P00352 4/20 0.49
TP53 P04637 1/20 0.49
DHFR P00374 3/20 0.45
KDM4E B2RXH2 4/20 0.45
SMN1; SMN2 Q16637 3/20 0.45
MAPT P10636 3/20 0.45
TUBB4A P04350 1/20 0.44
TUBB P07437 1/20 0.44
TUBA3C P0DPH7 1/20 0.44
TUBA1B P68363 1/20 0.44
TUBA4A P68366 1/20 0.44
TUBB4B P68371 1/20 0.44
TUBB3 Q13509 1/20 0.44
TUBB2A Q13885 1/20 0.44
TUBB8 Q3ZCM7 1/20 0.44
TUBA3E Q6PEY2 1/20 0.44
TUBA1A Q71U36 1/20 0.44
TUBA1C Q9BQE3 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6313851 1.00 KMT2A (0.51) KMT2AMEN1ALDH1A1TP53DHFR
SCHEMBL6306212 0.93 KMT2A (0.51) KMT2AMEN1ALDH1A1TP53DHFR
SCHEMBL6306210 0.93 KMT2A (0.51) KMT2AMEN1ALDH1A1TP53DHFR
SCHEMBL7554190 0.90 ALDH1A1 (0.55) KMT2AMEN1ALDH1A1TP53DHFR
SCHEMBL7554195 0.90 ALDH1A1 (0.55) KMT2AMEN1ALDH1A1TP53DHFR
SCHEMBL6313969 0.90 ALDH1A1 (0.58) KMT2AMEN1ALDH1A1TP53DHFR
SCHEMBL6313965 0.90 ALDH1A1 (0.58) KMT2AMEN1ALDH1A1TP53DHFR
SCHEMBL6309745 0.89 KMT2A (0.64) KMT2AMEN1ALDH1A1TP53KDM4E
SCHEMBL6309743 0.89 KMT2A (0.64) KMT2AMEN1ALDH1A1TP53KDM4E
SCHEMBL6307031 0.88 MEN1 (0.49) KMT2AMEN1ALDH1A1TP53DHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6890930-B1 Quinazolinones 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2005-05-10 US disclosed
EP-1216235-A1 QUINAZOLINONES MERCK PATENT GmbH (DE) 2002-06-26 EP disclosed
WO-2001023365-A1 QUINAZOLINONES MERCK PATENT GMBH (DE) 2001-04-05 WO disclosed