SCHEMBL6315148

SCHEMBL6315148

NCc1cccc(Cn2c(-c3ccc(-c4ccccc4)cc3)nc3cc(Cl)ccc3c2=O)c1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 4/20 0.66
ALDH1A1 P00352 7/20 0.61
SMN1; SMN2 Q16637 2/20 0.61
LMNA P02545 1/20 0.60
RECQL P46063 1/20 0.60
RAB9A P51151 1/20 0.60
MEN1 O00255 1/20 0.56
KMT2A Q03164 1/20 0.56
CYP1A2 P05177 1/20 0.55
GAA P10253 1/20 0.55
CYP2D6 P10635 1/20 0.55
CYP2C9 P11712 1/20 0.55
CYP2C19 P33261 1/20 0.55
F11 P03951 2/20 0.52
HTT P42858 1/20 0.51
BCL2 P10415 1/20 0.47
MCL1 Q07820 1/20 0.47
AVPR1B P47901 1/20 0.47
CASR P41180 1/20 0.46
KIF11 P52732 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6308313 0.98 EGFR (0.69) EGFRALDH1A1SMN1; SMN2LMNARECQL
SCHEMBL6308219 0.93 ALDH1A1 (0.60) EGFRALDH1A1SMN1; SMN2LMNARECQL
SCHEMBL6313535 0.92 ALDH1A1 (0.61) EGFRALDH1A1SMN1; SMN2LMNARECQL
SCHEMBL6308855 0.92 EGFR (0.59) EGFRALDH1A1SMN1; SMN2LMNARECQL
SCHEMBL6308153 0.90 ALDH1A1 (0.62) EGFRALDH1A1SMN1; SMN2LMNARECQL
SCHEMBL6309852 0.90 EGFR (0.55) EGFRALDH1A1SMN1; SMN2LMNARECQL
SCHEMBL6310387 0.90 EGFR (0.57) EGFRALDH1A1SMN1; SMN2LMNARECQL
SCHEMBL6306194 0.89 ALDH1A1 (0.72) EGFRALDH1A1SMN1; SMN2LMNARECQL
SCHEMBL6307768 0.88 EGFR (0.53) EGFRALDH1A1SMN1; SMN2LMNARECQL
SCHEMBL6314132 0.88 EGFR (0.53) EGFRALDH1A1SMN1; SMN2LMNARECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6890930-B1 Quinazolinones 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2005-05-10 US disclosed
EP-1216235-A1 QUINAZOLINONES MERCK PATENT GmbH (DE) 2002-06-26 EP disclosed
WO-2001023365-A1 QUINAZOLINONES MERCK PATENT GMBH (DE) 2001-04-05 WO disclosed