SCHEMBL631589

SCHEMBL631589

CC(C(Br)Br)N1CC(=O)NC1=O

nearest known ligand 0.48

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 3/20 0.48
TOP2B Q02880 3/20 0.48
ALDH1A1 P00352 1/20 0.48
MAPT P10636 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
CRBN Q96SW2 1/20 0.41
PTGS1 P23219 2/20 0.36
LMNA P02545 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL631865 0.84 TOP2A (0.45) TOP2ATOP2BALDH1A1MAPTTDP1
SCHEMBL29125125 0.83 TOP2A (0.46) TOP2ATOP2BALDH1A1MAPTTDP1
SCHEMBL630915 0.79 TOP2A (0.48) TOP2ATOP2BALDH1A1MAPTTDP1
SCHEMBL4971941 0.79 TOP2A (0.44) TOP2ATOP2BALDH1A1MAPTTDP1
SCHEMBL16597500 0.78 TOP2A (0.50) TOP2ATOP2BALDH1A1MAPTTDP1
SCHEMBL7823878 0.74 CRBN (0.39) TOP2ATOP2BALDH1A1MAPTTDP1
SCHEMBL11086765 0.74 TOP2A (0.46) TOP2ATOP2BALDH1A1MAPTTDP1
SCHEMBL10765254 0.74 TOP2A (0.46) TOP2ATOP2BALDH1A1MAPTTDP1
SCHEMBL27618934 0.74 TOP2A (0.46) TOP2ATOP2BALDH1A1MAPTTDP1
SCHEMBL11598867 0.73 CRBN (0.40) TOP2ATOP2BALDH1A1MAPTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 105 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2865743-B1 Improvements in dispensing devices RECKITT BENCKISER LLC (US) 2024-03-27 EP disclosed
EP-2952570-B1 IMPROVEMENTS IN DISPENSING DEVICES AND COMPOSITIONS THEREFOR RECKITT BENCKISER LLC (US) 2021-07-28 EP disclosed
EP-2191077-B1 CAGELESS DISPENSING DEVICE RECKITT BENCKISER LLC (US) 2017-03-15 EP disclosed
EP-3088616-A1 METHOD FOR PRODUCTION OF DISPENSING DEVICES Reckitt Benckiser LLC (US) 2016-11-02 EP disclosed
EP-2310583-B1 DISPENSING DEVICE FOR TOILET BOWL RECKITT BENCKISER LLC (US) 2016-10-05 EP disclosed
US-9334640-B2 Cageless dispensing device RECKITT BENCKISER LLC. (US) 2016-05-10 US disclosed
EP-1636437-B1 IMPROVED DISPENSING DEVICE RECKITT BENCKISER LLC (US) 2015-12-09 EP disclosed
EP-2952570-A1 IMPROVEMENTS IN DISPENSING DEVICES AND COMPOSITIONS THEREFOR Reckitt Benckiser LLC (US) 2015-12-09 EP disclosed
EP-1996691-B1 IMPROVEMENTS IN DISPENSING DEVICES RECKITT BENCKISER LLC (US) 2015-05-06 EP disclosed
EP-2865743-A1 Improvements in dispensing devices Reckitt Benckiser LLC (US) 2015-04-29 EP disclosed
WO-2004018581-A2 RESIN CURING AGENTS, COMPOSITIONS AND PRODUCTS CONTAINING SAME BIOLAB, INC. (US) 2004-03-04 WO disclosed
WO-2003042462-A2 IMPROVEMENTS RELATING TO TOILET BOWL CLEANING ARTICLES RECKITT BENCKISER INC (US) 2003-05-22 WO disclosed
US-6319356-B1 INHIBITING AUTOXIDATION OF UNSATURATED FATTY ACIDS AND/OR ESTERS IN PULP FIBER; OXIDIZATION BY ADDITION OF A HALOHYDANTOIN GREAT LAKES CHEMICAL CORPORATION 2001-11-20 US disclosed
EP-1095185-A4 PROCESS FOR CONTROLLING ODOR IN PAPER AND PAPERBOARD GREAT LAKES CHEMICAL CORP (US) 2001-10-17 EP disclosed
EP-1095185-A1 PROCESS FOR CONTROLLING ODOR IN PAPER AND PAPERBOARD GREAT LAKES CHEMICAL CORPORATION (US) 2001-05-02 EP disclosed
WO-1999058759-A1 PROCESS FOR CONTROLLING ODOR IN PAPER AND PAPERBOARD GREAT LAKES CHEMICAL CORPORATION (US) 1999-11-18 WO disclosed
US-5981461-A APPLYING TO THE OILY SURFACE AN AQUEOUS FLUID COMPRISING DIALKYLDIHALOHYDANTOIN AND A SULFONSUCCINATE SALT LONZA INC. (US) 1999-11-09 US disclosed
EP-0946694-A2 CLEANING COMPOSITIONS CONTAINING A HALOGEN BLEACHING AGENT AND A SULFOSUCCINATE SALT LONZA INC. (US) 1999-10-06 EP disclosed
WO-1998026033-A2 CLEANING COMPOSITIONS CONTAINING A HALOGEN BLEACHING AGENT AND A SULFOSUCCINATE SALT LONZA INC. (US) 1998-06-18 WO disclosed
US-4537697-A Method of enhancing solubility of halogenated hydantoins GLYCO, INC. (US) 1985-08-27 US disclosed