SCHEMBL6320052

SCHEMBL6320052

Cc1ccccc1-c1ccsc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 5/20 0.52
CYP2B6 P20813 3/20 0.52
CYP2E1 P05181 1/20 0.52
PTPRC P08575 1/20 0.44
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
MAOB P27338 1/20 0.41
EDNRA P25101 1/20 0.40
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40
TP53 P04637 1/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
GPR35 Q9HC97 1/20 0.39
TDO2 P48775 1/20 0.39
ADRA2A P08913 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1132878 0.84 CYP2A6 (0.45) CYP2A6CYP2B6CYP2E1PTPRCCYP3A4
SCHEMBL4946960 0.84 CYP2A6 (0.64) CYP2A6CYP2B6CYP2E1PTPRCCYP3A4
SCHEMBL27465618 0.83 PDCD1 (0.44) CYP2A6CYP2B6CYP2E1PTPRCCYP3A4
SCHEMBL2094933 0.82 CYP2A6 (0.42) CYP2A6CYP2B6CYP2E1PTPRCCYP3A4
SCHEMBL7058734 0.77 CYP2A6 (0.70) CYP2A6CYP2B6CYP2E1PTPRCCYP3A4
SCHEMBL21848864 0.76 CYP2A6 (0.59) CYP2A6CYP2B6CYP2E1CYP3A4CYP2C9
SCHEMBL3181535 0.76 CYP2A6 (0.54) CYP2A6CYP2B6CYP2E1PTPRCCYP3A4
SCHEMBL27870289 0.76 CYP2A6 (0.67) CYP2A6CYP2B6CYP2E1PTPRCCYP3A4
SCHEMBL21562299 0.75 CYP2A6 (0.42) CYP2A6CYP2B6CYP3A4CYP2C9CYP2C19
SCHEMBL14003393 0.75 CYP2A6 (0.53) CYP2A6CYP2B6CYP2E1CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113264816-B Spiro [ cyclopropane-1, 2' -indene ] -1',3' -diketone derivative and synthetic method thereof 湖北科技学院 2023-03-24 CN disclosed
WO-2020018747-A1 METHOD OF MODULATING RIBONUCLEOTIDE REDUCTASE CASE WESTERN RESERVE UNIVERSITY (US) 2020-01-23 WO disclosed
WO-2017121969-A1 NOVEL PHOSPHINANE AND AZAPHOSPHINANE DERIVATIVES, METHOD FOR PREPARING SAME AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME LES LABORATOIRES SERVIER (FR) 2017-07-20 WO disclosed
CN-104529850-A Method for preparing (Z) type tellurium-sulfur olefin compound UNIV HUNAN 2015-04-22 CN disclosed
US-7271270-B2 High affinity small molecule C5a receptor modulators NEUROGEN CORPORATION (US) 2007-09-18 US disclosed
CN-1280300-C Heterocyclic metallocene compounds and use thereof in catalyst systems for producing olefin polymers BASELL TECHNOLOGY CO BV (NL) 2006-10-18 CN disclosed
US-6924301-B1 Composition for treating or preventing arrhythmia SHIONOGI & CO., LTD. (JP) 2005-08-02 US disclosed
CN-1161388-C Metallocene compounds, process for their preparation and their use in catalytic systems for polymerization of olefins 2004-08-11 CN disclosed
EP-0976748-B1 PYRROLIDINE DERIVATIVES HAVING PHOSPHOLIPASE A2 INHIBITORY ACTIVITY SHIONOGI & CO (JP) 2003-12-03 EP disclosed
EP-1240906-A1 PREVENTIVES OR REMEDIES FOR ARRHYTHMIA SHIONOGI & CO., LTD. (JP) 2002-09-18 EP disclosed
CN-1348459-A Heterocyclic metallocene compounds and their use in catalyst systems for producing olefin polymers BASELL TECHNOLOGY CO BV (NL) 2002-05-08 CN disclosed
CN-1347424-A Metallocene compounds, process for their preparation and their use in catalytic systems for polymerization of olefins BASELL TECHNOLOGY CO B V (NL) 2002-05-01 CN disclosed
US-6147100-A ANTIINFLAMMATORY AGENTS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
EP-0976748-A1 PYRROLIDINE DERIVATIVES HAVING PHOSPHOLIPASE A2 INHIBITORY ACTIVITY SHIONOGI & CO., LTD. (JP) 2000-02-02 EP disclosed
US-4599341-A CARDIOVASCULAR DISORDERS MERCK & CO., INC. (US) 1986-07-08 US disclosed