SCHEMBL4946960

SCHEMBL4946960

c1ccc(-c2ccsc2)c(-c2ccsc2)c1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 4/20 0.64
CYP2B6 P20813 2/20 0.64
CYP2E1 P05181 1/20 0.64
PTPRC P08575 1/20 0.52
CYP3A4 P08684 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50
MAOB P27338 1/20 0.47
TDO2 P48775 1/20 0.45
PDGFRB P09619 1/20 0.42
PDGFRA P16234 1/20 0.42
PDK2 Q15119 1/20 0.42
ADRA1D P25100 1/20 0.41
ADRA1A P35348 1/20 0.41
ADRA1B P35368 1/20 0.41
KCNH2 Q12809 1/20 0.41
NQO2 P16083 1/20 0.41
CDK8 P49336 1/20 0.41
GPR84 Q9NQS5 1/20 0.40
ADRA2A P08913 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7058734 0.93 CYP2A6 (0.70) CYP2A6CYP2B6CYP2E1PTPRCCYP3A4
SCHEMBL27870289 0.91 CYP2A6 (0.67) CYP2A6CYP2B6CYP2E1PTPRCCYP3A4
SCHEMBL3181535 0.85 CYP2A6 (0.54) CYP2A6CYP2B6CYP2E1PTPRCCYP3A4
SCHEMBL26259978 0.84 CYP2A6 (0.58) CYP2A6CYP2B6CYP2E1PTPRCCYP3A4
SCHEMBL26259994 0.84 CYP2A6 (0.52) CYP2A6CYP2B6CYP2E1PTPRCCYP3A4
SCHEMBL1310377 0.84 ALDH1A1 (0.54) CYP2A6CYP2B6CYP2E1PTPRCCYP3A4
SCHEMBL7744328 0.84 CYP2A6 (0.52) CYP2A6CYP2B6CYP2E1PTPRCCYP3A4
SCHEMBL6829969 0.84 CYP2A6 (0.52) CYP2A6CYP2B6CYP2E1PTPRCCYP3A4
SCHEMBL1309148 0.84 CYP2A6 (0.54) CYP2A6CYP2B6CYP2E1PTPRCCYP3A4
SCHEMBL3240839 0.84 CYP2A6 (0.52) CYP2A6CYP2B6CYP2E1PTPRCCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080188670-A1 1,4-Dithienylbenzene Derivative NAT. INST. OF ADVANCED INDUSTRIAL SCI. AND TECH. (JP) 2008-08-07 US claimed
CN-108191817-A The activity of the resisting tobacco mosaic virus of the 2- methyl butyne amine acylated derivatives of the dithienyl benzene structure containing 1,3- 南开大学 2018-06-22 CN disclosed
CN-104973805-A conductive polymer-graphene composite electrochromic film and preparation method thereof UNIV ZHEJIANG TECHNOLOGY 2015-10-14 CN disclosed
WO-2013009032-A2 NOVEL ORGANIC ELECTROLUMINESCENT COMPOUND, AND ORGANIC ELECTROLUMINESCENT DEVICE INCLUDING SAME 주식회사 두산 (KR) 2013-01-17 WO disclosed
US-20080188670-A1 1,4-Dithienylbenzene Derivative NAT. INST. OF ADVANCED INDUSTRIAL SCI. AND TECH. (JP) 2008-08-07 US disclosed
US-20080188670-A1 1,4-Dithienylbenzene Derivative NAT. INST. OF ADVANCED INDUSTRIAL SCI. AND TECH. (JP) 2008-08-07 US disclosed
US-20080188670-A1 1,4-Dithienylbenzene Derivative NAT. INST. OF ADVANCED INDUSTRIAL SCI. AND TECH. (JP) 2008-08-07 US disclosed
JP-2007059558-A ORGANIC SEMICONDUCTOR ELEMENT NATIONAL INSTITUTE OF ADVANCED INDUSTRIAL & TECHNOLOGY 2007-03-08 JP disclosed
WO-2006022040-A1 1,4-DITHIENYLBENZENE DERIVATIVE NATIONAL INSTITUTE OF ADVANCED INDUSTRIAL SCIENCE AND TECHNOLOGY (JP) 2006-03-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080188670-A1 1,4-Dithienylbenzene Derivative SLC22A4, SLC19A2, SLC22A1 CYP2A6 3908/4885CYP2B6 2375/4885CYP2E1 661/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.