SCHEMBL6325693

SCHEMBL6325693

C=CC(=O)NC1CCCC(Nc2n[nH]c(=O)c3cccnc23)C1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BTK Q06187 5/20 0.45
KCNH2 Q12809 1/20 0.45
JAK3 P52333 4/20 0.41
ROCK2 O75116 2/20 0.39
CDC7 O00311 2/20 0.39
DAPK3 O43293 2/20 0.39
MAP4K4 O95819 2/20 0.39
PAK4 O96013 2/20 0.39
PIM1 P11309 2/20 0.39
PRKACA P17612 2/20 0.39
CDK2 P24941 2/20 0.39
FLT3 P36888 2/20 0.39
CSNK1A1 P48729 2/20 0.39
CLK2 P49760 2/20 0.39
GSK3B P49841 2/20 0.39
CDK7 P50613 2/20 0.39
CDK9 P50750 2/20 0.39
PRKX P51817 2/20 0.39
CDK5 Q00535 2/20 0.39
MAP4K2 Q12851 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6324540 0.87 JAK3 (0.48) BTKJAK3ROCK2CDC7DAPK3
SCHEMBL6326421 0.87 BTK (0.48) BTKKCNH2JAK3ROCK2GRM5
SCHEMBL5076306 0.84 ROCK2 (0.45) JAK3ROCK2CDC7DAPK3MAP4K4
SCHEMBL6327186 0.82 CD38 (0.41) ROCK2ROCK1PARP1GRM4JAK2
SCHEMBL6325411 0.80 BRD4 (0.48) BTKJAK3ROCK2CDC7DAPK3
SCHEMBL6325659 0.80 BRD4 (0.48) BTKJAK3ROCK2CDC7DAPK3
SCHEMBL6325665 0.80 BRD4 (0.48) BTKJAK3ROCK2CDC7DAPK3
SCHEMBL6326484 0.79 JAK3 (0.48) BTKJAK3ROCK2CDC7DAPK3
SCHEMBL6328374 0.77 ROCK2 (0.42) JAK3ROCK2CDC7DAPK3MAP4K4
SCHEMBL6328383 0.73 ROCK2 (0.48) BTKJAK3ROCK2CDC7DAPK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6924284-B2 PARP inhibitors ICOS CORPORATION (US) 2005-08-02 US disclosed