SCHEMBL6340487

SCHEMBL6340487

CCOCCOc1ccc(-c2ccc3c(c2)C=C(C(=O)Nc2ccc(CN(C)C4CCOCC4)cc2)CCN3S(C)(=O)=O)cc1

nearest known ligand 0.56

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 4/20 0.56
CCR5 P51681 16/20 0.46
CCR3 P51677 1/20 0.42
CCR4 P51679 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6343618 0.97 CCR2 (0.56) CCR2CCR5CCR3CCR4MEN1
SCHEMBL6429556 0.94 CCR2 (0.56) CCR2CCR5CCR3CCR4MEN1
SCHEMBL6349106 0.94 CCR2 (0.57) CCR2CCR5MEN1KMT2A
SCHEMBL6342643 0.92 CCR2 (0.54) CCR2CCR5CCR3CCR4
SCHEMBL6349220 0.91 CCR2 (0.54) CCR2CCR5MEN1KMT2A
SCHEMBL3038176 0.91 CCR2 (0.58) CCR2CCR5CCR3CCR4
SCHEMBL6343858 0.91 CCR2 (0.58) CCR2CCR5
SCHEMBL6344086 0.90 CCR2 (0.57) CCR2CCR5CCR3CCR4MEN1
SCHEMBL3026515 0.89 CCR2 (0.56) CCR2CCR5
SCHEMBL6351851 0.88 CCR2 (0.58) CCR2CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6936602-B1 Benzazepine derivatives, process for the preparation of the same and uses thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2005-08-30 US disclosed
EP-1186604-A1 BENZAZEPINE DERIVATIVES, PROCESS FOR THE PREPARATION OF THE SAME AND USES THEREOF Takeda Chemical Industries, Ltd. (JP) 2002-03-13 EP disclosed