SCHEMBL6344879

SCHEMBL6344879

CCCCOCCOc1ccc(-c2ccc3c(c2)C=C(C(=O)Nc2ccc(CN(C)C4CCOCC4)cc2)CCN3c2ccc(S(N)(=O)=O)cc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 5/20 0.49
CCR5 P51681 17/20 0.45
CCR3 P51677 1/20 0.43
CCR4 P51679 1/20 0.43
CCR7 P32248 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6351882 0.94 CCR2 (0.49) CCR2CCR5CCR3CCR4CCR7
SCHEMBL6412038 0.94 CCR2 (0.49) CCR2CCR5CCR3CCR4CCR7
SCHEMBL6341719 0.93 CCR2 (0.53) CCR2CCR5CCR3CCR4CCR7
SCHEMBL6340444 0.92 CCR2 (0.52) CCR2CCR5CCR3CCR4CCR7
SCHEMBL3037836 0.92 CCR2 (0.53) CCR2CCR5CCR3CCR4CCR7
SCHEMBL6151154 0.89 CCR2 (0.50) CCR2CCR5CCR3CCR4CCR7
SCHEMBL6342683 0.89 CCR2 (0.51) CCR2CCR5CCR3CCR4CCR7
Hydrochloric Acid SCHEMBL6350708 0.89 CCR2 (0.52) CCR2CCR5CCR3CCR4CCR7
SCHEMBL6342835 0.87 CCR2 (0.52) CCR2CCR5CCR3CCR4CCR7
SCHEMBL6343762 0.87 CCR2 (0.56) CCR2CCR5CCR3CCR4CCR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6936602-B1 Benzazepine derivatives, process for the preparation of the same and uses thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2005-08-30 US disclosed
EP-1186604-A1 BENZAZEPINE DERIVATIVES, PROCESS FOR THE PREPARATION OF THE SAME AND USES THEREOF Takeda Chemical Industries, Ltd. (JP) 2002-03-13 EP disclosed