SCHEMBL6345215

SCHEMBL6345215

Oc1ccc2c(c1O)Oc1cccc3c1C2CNC3

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.46
CYP3A4 P08684 5/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
CYP2D6 P10635 1/20 0.39
PARP1 P09874 1/20 0.39
DRD2 P14416 2/20 0.38
DRD1 P21728 2/20 0.38
MAPK1 P28482 4/20 0.33
HSD17B10 Q99714 4/20 0.33
ALOX15 P16050 2/20 0.33
TSHR P16473 2/20 0.33
NFKB1 P19838 2/20 0.33
THPO P40225 2/20 0.33
KDM4E B2RXH2 5/20 0.33
MAPT P10636 5/20 0.33
HPGD P15428 5/20 0.33
ALDH1A1 P00352 3/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
LMNA P02545 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29383649 1.00 HTR2A (0.46) HTR2ACYP3A4MEN1KMT2ACYP2D6
Bromide SCHEMBL3668719 0.99 HTR2A (0.45) HTR2ACYP3A4MEN1KMT2ACYP2D6
SCHEMBL22952971 0.84 HTR2A (0.35) HTR2ACYP3A4MEN1KMT2ACYP2D6
SCHEMBL22953341 0.78 PARP1 (0.43) CYP3A4MEN1KMT2ACYP2D6PARP1
SCHEMBL6391686 0.77 HTR2A (0.60) HTR2ACYP3A4MEN1KMT2ACYP2D6
SCHEMBL3680945 0.75 HTR2A (0.42) HTR2ACYP3A4MEN1KMT2ACYP2D6
SCHEMBL22952976 0.74 HTR2A (0.33) HTR2ACYP3A4MEN1KMT2ACYP2D6
SCHEMBL16938669 0.74 HTR2A (0.60) HTR2ACYP3A4MEN1KMT2ACYP2D6
SCHEMBL29383346 0.74 HTR2A (0.60) HTR2ACYP3A4MEN1KMT2ACYP2D6
SCHEMBL3672464 0.74 HTR2A (0.60) HTR2ACYP3A4MEN1KMT2ACYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050232870-A1 Method of treatment of dopamine-related dysfunction PURDUE RESEARCH FOUNDATION AND UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL 2005-10-20 US disclosed
US-6916823-B2 Method of treatment of dopamine-related dysfunction PURDUE RESEARCH FOUNDATION (US) 2005-07-12 US disclosed
US-20050080266-A1 CHROMENO[4,3,2-DE]ISOQUINOLINES AS POTENT DOPAMINE RECEPTOR LIGANDS NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2005-04-14 US disclosed
US-6413977-B1 D1 AGONISTS; CENTRAL AND PERIPHERAL NERVOUS SYSTEM DYSFUNCTIONS; IMPROVING COGNITION AND MEMORY; PARKINSON'S DISEASE, SCHIZOPHRENIA, ATTENTION-DEFICIT HYPERACTIVITY, SUBSTANCE ABUSE, PHYSIOLOGICAL FUNCTION PURDUE RESEARCH FOUNDATION 2002-07-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050232870-A1 Method of treatment of dopamine-related dysfunction DRD2, DRD1, DRD3 HTR2A 43/4885CYP3A4 694/4885MEN1 3521/4885
US-20050080266-A1 CHROMENO[4,3,2-DE]ISOQUINOLINES AS POTENT DOPAMINE RECEPTOR LIGANDS DRD2, COMT, CHRM3 HTR2A 22/4885CYP3A4 210/4885MEN1 4885/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.