SCHEMBL6350345

SCHEMBL6350345

CCCOC(C)Oc1ccc(-c2ccc3c(c2)C=C(C(=O)Nc2ccc(CN(C)C4CCOCC4)cc2)CCN3Cc2cccs2)cc1

nearest known ligand 0.49

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 4/20 0.49
CCR5 P51681 16/20 0.44
CCR7 P32248 1/20 0.37
CXCR5 P32302 1/20 0.36
CXCR3 P49682 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6350462 0.97 CCR2 (0.49) CCR2CCR5CCR7CXCR5CXCR3
SCHEMBL6339026 0.91 CCR2 (0.55) CCR2CCR5CCR7CXCR3
SCHEMBL6351375 0.91 CCR2 (0.49) CCR2CCR5CCR7CXCR3
SCHEMBL6350252 0.90 CCR2 (0.52) CCR2CCR5CCR7CXCR3
SCHEMBL6350338 0.89 CCR2 (0.51) CCR2CCR5CCR7
SCHEMBL6349394 0.89 CCR2 (0.51) CCR2CCR5CCR7
SCHEMBL6339060 0.89 CCR2 (0.49) CCR2CCR5CCR7CXCR5CXCR3
SCHEMBL6341920 0.89 CCR2 (0.51) CCR2CCR5CCR7CXCR5CXCR3
SCHEMBL6339034 0.88 CCR2 (0.48) CCR2CCR5CCR7CXCR5CXCR3
SCHEMBL6350458 0.88 CCR2 (0.51) CCR2CCR5CCR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6936602-B1 Benzazepine derivatives, process for the preparation of the same and uses thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2005-08-30 US disclosed
EP-1186604-A1 BENZAZEPINE DERIVATIVES, PROCESS FOR THE PREPARATION OF THE SAME AND USES THEREOF Takeda Chemical Industries, Ltd. (JP) 2002-03-13 EP disclosed