SCHEMBL6358019

SCHEMBL6358019

CCOc1ccc(C#Cc2ccc(OC)cc2C=O)cc1

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 3/20 0.46
ALDH1A1 P00352 1/20 0.43
KDM4E B2RXH2 1/20 0.43
RAB9A P51151 1/20 0.43
ESR1 P03372 2/20 0.42
AHR P35869 1/20 0.42
TRIM24 O15164 1/20 0.42
TYR P14679 1/20 0.42
TRIM33 Q9UPN9 1/20 0.42
ACACB O00763 11/20 0.41
NQO1 P15559 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9881727 0.90 ERN1 (0.51) ERN1ALDH1A1KDM4ETRIM24TYR
SCHEMBL4765815 0.84 ERN1 (0.49) ERN1ALDH1A1KDM4ERAB9ATRIM24
SCHEMBL6358014 0.83 ALDH1A1 (0.43) ERN1ALDH1A1KDM4ERAB9ATRIM24
SCHEMBL7601226 0.80 APP (0.44) ERN1ALDH1A1TRIM24TYRTRIM33
SCHEMBL18641647 0.77 ERN1 (0.47) ERN1ALDH1A1KDM4ERAB9ATRIM24
SCHEMBL3612866 0.76 ERN1 (0.44) ERN1ALDH1A1KDM4EACACB
SCHEMBL312237 0.75 ALDH1A1 (0.53) ERN1ALDH1A1RAB9ATRIM24TYR
SCHEMBL30134856 0.75 ALDH1A1 (0.53) ERN1ALDH1A1RAB9ATRIM24TYR
SCHEMBL4770355 0.74 ALDH1A1 (0.53) ERN1ALDH1A1TRIM24TYRTRIM33
SCHEMBL20488634 0.74 KDM4E (0.59) ERN1ALDH1A1KDM4ERAB9ATRIM24

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6875761-B2 Certain 1,3-disubstituted isoquinoline derivatives EISAI CO., LTD. (JP) 2005-04-05 US disclosed