SCHEMBL6367392

SCHEMBL6367392

CC(C)(C)Oc1ccc(C[C@H](NC(=O)[C@@H]2CCCN2S(=O)(=O)c2ccc(S(=O)(=O)c3ccc(C(F)(F)F)cc3)s2)C(=O)O)cc1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 10/20 0.46
ITGA5 P08648 3/20 0.46
ITGA4 P13612 5/20 0.46
ITGB7 P26010 1/20 0.46
KCNQ1 P51787 1/20 0.43
TRPA1 O75762 1/20 0.43
HCRTR1 O43613 3/20 0.42
HCRTR2 O43614 3/20 0.42
ITGAV P06756 4/20 0.41
BRD4 O60885 1/20 0.41
KDM4E B2RXH2 1/20 0.40
KDM4A O75164 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6367886 0.92 ITGB1 (0.55) ITGB1ITGA5ITGA4ITGB7HCRTR1
SCHEMBL6367319 0.82 ITGB1 (0.53) ITGB1ITGA5ITGA4ITGB7KCNQ1
SCHEMBL6368426 0.81 ITGB1 (0.58) ITGB1ITGA5ITGA4ITGB7HCRTR1
SCHEMBL6431309 0.81 ITGB1 (0.58) ITGB1ITGA5ITGA4ITGB7HCRTR1
SCHEMBL6429378 0.81 ITGB1 (0.67) ITGB1ITGA5ITGA4ITGB7ITGAV
SCHEMBL6367276 0.81 ITGB1 (0.48) ITGB1ITGA5ITGA4ITGB7HCRTR1
SCHEMBL6373924 0.81 ITGB1 (0.59) ITGB1ITGA5ITGA4ITGB7HCRTR1
SCHEMBL6373884 0.79 ITGB1 (0.45) ITGB1ITGA5ITGA4ITGB7TRPA1
SCHEMBL6367527 0.78 ITGB1 (0.71) ITGB1ITGA5ITGA4ITGB7ITGAV
SCHEMBL6369020 0.76 ITGB1 (0.57) ITGB1ITGA5ITGA4ITGB7HCRTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001764-A4 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO INC (US) 2005-08-24 EP claimed
US-6903075-B1 Heterocyclic amide compounds as cell adhesion inhibitors MERCK & CO., INC. (US) 2005-06-07 US claimed
JP-2002512625-A 2002-04-23 JP claimed
EP-1001764-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS Merck & Co., Inc. (a New Jersey corp.) (US) 2000-05-24 EP claimed
WO-1999064395-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1999-12-16 WO claimed
WO-1998053814-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1998-12-03 WO claimed