SCHEMBL6367276

SCHEMBL6367276

CC(C)(C)Oc1ccc(C[C@H](NC(=O)[C@@H]2CCCN2S(=O)(=O)c2ccc(CNC(=O)c3ccccc3)s2)C(=O)O)cc1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 10/20 0.48
ITGA5 P08648 4/20 0.48
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
ITGA4 P13612 6/20 0.46
ITGB7 P26010 1/20 0.46
ITGA2 P17301 1/20 0.43
ITGAV P06756 3/20 0.42
ACE P12821 1/20 0.41
ITGB3 P05106 1/20 0.41
CACNA1B Q00975 1/20 0.40
USP2 O75604 1/20 0.40
GAA P10253 1/20 0.40
HCRTR1 O43613 1/20 0.40
HCRTR2 O43614 1/20 0.40
CMA1 P23946 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7450243 0.88 ITGB1 (0.51) ITGB1ITGA5MEN1KMT2AITGA4
SCHEMBL6367886 0.86 ITGB1 (0.55) ITGB1ITGA5ITGA4ITGB7ITGA2
SCHEMBL6429378 0.83 ITGB1 (0.67) ITGB1ITGA5ITGA4ITGB7ITGA2
SCHEMBL6367392 0.81 ITGB1 (0.46) ITGB1ITGA5ITGA4ITGB7ITGAV
SCHEMBL6367319 0.79 ITGB1 (0.53) ITGB1ITGA5MEN1KMT2AITGA4
SCHEMBL6429533 0.79 ITGB1 (0.52) ITGB1ITGA5ITGA4ITGB7ITGA2
SCHEMBL6368426 0.78 ITGB1 (0.58) ITGB1ITGA5ITGA4ITGB7USP2
SCHEMBL6431309 0.78 ITGB1 (0.58) ITGB1ITGA5KMT2AITGA4ITGB7
SCHEMBL6367527 0.77 ITGB1 (0.71) ITGB1ITGA5ITGA4ITGB7ITGAV
SCHEMBL6368567 0.77 ITGB1 (0.55) ITGB1ITGA5ITGA4ITGB7ITGA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001764-A4 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO INC (US) 2005-08-24 EP claimed
US-6903075-B1 Heterocyclic amide compounds as cell adhesion inhibitors MERCK & CO., INC. (US) 2005-06-07 US claimed
JP-2002512625-A 2002-04-23 JP claimed
EP-1001764-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS Merck & Co., Inc. (a New Jersey corp.) (US) 2000-05-24 EP claimed
WO-1999064395-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1999-12-16 WO claimed
WO-1998053814-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1998-12-03 WO claimed