SCHEMBL6368246

SCHEMBL6368246

O=C(O)C[C@H](NC(=O)[C@@H]1CCCN1S(=O)(=O)c1cc(Cl)cc(Cl)c1)C(=O)O

nearest known ligand 0.73

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 20/20 0.73
ITGA4 P13612 20/20 0.73
ITGB7 P26010 2/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7237195 0.90 ITGB1 (0.68) ITGB1ITGA4ITGB7
SCHEMBL6375057 0.89 ITGB1 (0.65) ITGB1ITGA4ITGB7
SCHEMBL6367743 0.89 ITGB1 (0.64) ITGB1ITGA4ITGB7
Hydrochloric Acid SCHEMBL6149929 0.88 ITGB1 (0.63) ITGB1ITGA4ITGB7
Hydrochloric Acid SCHEMBL6149933 0.88 ITGB1 (0.63) ITGB1ITGA4ITGB7
SCHEMBL7226827 0.86 ITGB1 (0.61) ITGB1ITGA4ITGB7
SCHEMBL6368512 0.85 ITGA4 (0.72) ITGB1ITGA4ITGB7
SCHEMBL6372412 0.85 ITGA4 (0.72) ITGB1ITGA4ITGB7
SCHEMBL6367973 0.85 ITGB1 (0.62) ITGB1ITGA4ITGB7
SCHEMBL6368456 0.84 ITGA4 (0.70) ITGB1ITGA4ITGB7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001764-A4 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO INC (US) 2005-08-24 EP claimed
US-6903075-B1 Heterocyclic amide compounds as cell adhesion inhibitors MERCK & CO., INC. (US) 2005-06-07 US claimed
JP-2002512625-A 2002-04-23 JP claimed
EP-1001764-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS Merck & Co., Inc. (a New Jersey corp.) (US) 2000-05-24 EP claimed
WO-1999064395-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1999-12-16 WO claimed
WO-1998053814-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1998-12-03 WO claimed