SCHEMBL6368448

SCHEMBL6368448

Cc1cccc(CC(NC(=O)[C@@H]2CCCN2S(=O)(=O)c2ccccc2)C(=O)O)c1

nearest known ligand 0.65

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 11/20 0.65
ITGA5 P08648 5/20 0.65
ITGA4 P13612 6/20 0.63
ITGA2 P17301 1/20 0.63
ALDH1A1 P00352 1/20 0.56
FKBP1A P62942 3/20 0.54
ITGAV P06756 3/20 0.54
ITGB7 P26010 2/20 0.52
ITGB3 P05106 1/20 0.51
MMP2 P08253 1/20 0.50
MMP9 P14780 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6368450 1.00 ITGB1 (0.65) ITGB1ITGA5ITGA4ITGA2ALDH1A1
SCHEMBL2879404 0.90 ITGB1 (0.77) ITGB1ITGA5ITGA4ITGA2ALDH1A1
SCHEMBL2879401 0.90 ITGB1 (0.77) ITGB1ITGA5ITGA4ITGA2ALDH1A1
SCHEMBL27877728 0.90 ITGB1 (0.77) ITGB1ITGA5ITGA4ITGA2ALDH1A1
SCHEMBL2879402 0.90 ITGB1 (0.77) ITGB1ITGA5ITGA4ITGA2ALDH1A1
SCHEMBL6710892 0.89 ALDH1A1 (0.70) ITGB1ITGA5ITGA4ITGA2ALDH1A1
SCHEMBL7066469 0.89 ALDH1A1 (0.70) ITGB1ITGA5ITGA4ITGA2ALDH1A1
SCHEMBL7069740 0.89 ALDH1A1 (0.70) ITGB1ITGA5ITGA4ITGA2ALDH1A1
SCHEMBL27514023 0.89 ALDH1A1 (0.70) ITGB1ITGA5ITGA4ITGA2ALDH1A1
SCHEMBL6439213 0.89 ALDH1A1 (0.70) ITGB1ITGA5ITGA4ITGA2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001764-A4 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO INC (US) 2005-08-24 EP claimed
US-6903075-B1 Heterocyclic amide compounds as cell adhesion inhibitors MERCK & CO., INC. (US) 2005-06-07 US claimed
JP-2002512625-A 2002-04-23 JP claimed
EP-1001764-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS Merck & Co., Inc. (a New Jersey corp.) (US) 2000-05-24 EP claimed
WO-1999064395-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1999-12-16 WO claimed
WO-1998053814-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1998-12-03 WO claimed
EP-1001764-A4 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO INC (US) 2005-08-24 EP disclosed
US-6903075-B1 Heterocyclic amide compounds as cell adhesion inhibitors MERCK & CO., INC. (US) 2005-06-07 US disclosed
EP-1001764-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS Merck & Co., Inc. (a New Jersey corp.) (US) 2000-05-24 EP disclosed
WO-1999064395-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1999-12-16 WO disclosed
WO-1998053814-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1998-12-03 WO disclosed