SCHEMBL6374167

SCHEMBL6374167

NS(=O)(=O)c1ccccc1-c1ccc(NC(=O)[C@@H](Cc2ccccc2)NC(=O)Nc2ccc(Cl)cc2)cc1

nearest known ligand 0.64

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
F10 P00742 8/20 0.64
SMN1; SMN2 Q16637 1/20 0.54
CA12 O43570 1/20 0.52
CA1 P00915 1/20 0.52
CA2 P00918 1/20 0.52
CA9 Q16790 1/20 0.52
PRSS1 P07477 4/20 0.48
F2 P00734 1/20 0.48
F9 P00740 1/20 0.48
PRSS2 P07478 1/20 0.48
PRSS3 P35030 1/20 0.48
FPR2 P25090 6/20 0.47
NAMPT P43490 1/20 0.46
ADAMTS5 Q9UNA0 1/20 0.46
MMP2 P08253 1/20 0.46
PLG P00747 1/20 0.46
PROC P04070 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6374177 1.00 F10 (0.64) F10SMN1; SMN2CA12CA1CA2
SCHEMBL6374977 0.90 F10 (0.52) F10SMN1; SMN2CA12CA1CA2
SCHEMBL6374974 0.90 F10 (0.52) F10SMN1; SMN2CA12CA1CA2
SCHEMBL6379420 0.90 F10 (0.52) F10SMN1; SMN2CA12CA1CA2
SCHEMBL6375154 0.90 F10 (0.55) F10SMN1; SMN2CA12CA1CA2
SCHEMBL6375140 0.87 USP30 (0.56) F10FPR2
SCHEMBL6381183 0.87 USP30 (0.56) F10FPR2
SCHEMBL6374070 0.84 F10 (0.55) F10SMN1; SMN2CA12CA1CA2
SCHEMBL6374074 0.84 F10 (0.55) F10SMN1; SMN2CA12CA1CA2
SCHEMBL6380705 0.84 F10 (0.55) F10SMN1; SMN2CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050137230-A1 Carboxamide derivatives DORSCH DIETER (DE) 2005-06-23 US claimed
US-20040038858-A1 Carboxamide derivatives and their use in the treatment of thromboembolic diseases and tumours MERCK PATENT GMBH (DE) 2004-02-26 US claimed
US-20050137230-A1 Carboxamide derivatives DORSCH DIETER (DE) 2005-06-23 US disclosed
US-20040038858-A1 Carboxamide derivatives and their use in the treatment of thromboembolic diseases and tumours MERCK PATENT GMBH (DE) 2004-02-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050137230-A1 Carboxamide derivatives F11, F12, F2 F10 4/4885SMN1; SMN2 2974/4885CA12 1466/4885
US-20040038858-A1 Carboxamide derivatives and their use in the treatment of thromboembolic diseases and tumours CNR2, CNR1, HCAR2 F10 117/4885SMN1; SMN2 3253/4885CA12 879/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.