SCHEMBL6374288

SCHEMBL6374288

O=C(O)[C@H](Cc1ccc2ccccc2c1)NC(=O)[C@@H]1CCCN1S(=O)(=O)c1cccc(Cl)c1

nearest known ligand 0.68

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 11/20 0.68
ITGA4 P13612 6/20 0.68
ITGB7 P26010 3/20 0.62
ITGA5 P08648 4/20 0.59
CCR4 P51679 3/20 0.53
HCRTR1 O43613 2/20 0.50
HCRTR2 O43614 2/20 0.50
ITGA2 P17301 1/20 0.49
ITGAV P06756 2/20 0.49
CAPN1 P07384 1/20 0.47
TACR1 P25103 1/20 0.47
LMNA P02545 1/20 0.47
HPGD P15428 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6368803 0.93 ITGB1 (0.68) ITGB1ITGA4ITGB7ITGA5CCR4
SCHEMBL6428866 0.92 ITGB1 (0.68) ITGB1ITGA4ITGB7ITGA5CCR4
SCHEMBL6368888 0.91 ITGB1 (0.73) ITGB1ITGA4ITGB7ITGA5HCRTR1
SCHEMBL6368166 0.88 ITGB1 (0.72) ITGB1ITGA4ITGB7ITGA5HCRTR1
SCHEMBL6373490 0.86 ITGB1 (0.66) ITGB1ITGA4ITGB7ITGA5HCRTR1
SCHEMBL7070076 0.86 CCR4 (0.64) ITGB1ITGA4ITGB7ITGA5CCR4
SCHEMBL7066228 0.86 ITGB1 (0.61) ITGB1ITGA4ITGB7ITGA5CCR4
SCHEMBL6368039 0.85 ITGB1 (0.66) ITGB1ITGA4ITGB7ITGA5HCRTR1
SCHEMBL6368508 0.84 ITGB1 (0.69) ITGB1ITGA4ITGB7ITGA5CCR4
SCHEMBL6373361 0.84 ITGB1 (0.56) ITGB1ITGA4ITGB7ITGA5CCR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001764-A4 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO INC (US) 2005-08-24 EP claimed
US-6903075-B1 Heterocyclic amide compounds as cell adhesion inhibitors MERCK & CO., INC. (US) 2005-06-07 US claimed
JP-2002512625-A 2002-04-23 JP claimed
EP-1001764-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS Merck & Co., Inc. (a New Jersey corp.) (US) 2000-05-24 EP claimed
WO-1999064395-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1999-12-16 WO claimed
WO-1998053814-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1998-12-03 WO claimed