SCHEMBL6374348

SCHEMBL6374348

Cn1cc(-c2ccccc2[N+](=O)[O-])cn1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.54
TDP1 Q9NUW8 1/20 0.54
BRD4 O60885 1/20 0.50
ERN1 O75460 1/20 0.48
SMARCA2 P51531 1/20 0.44
SMARCA4 P51532 1/20 0.44
ADRA1A P35348 2/20 0.42
PDK2 Q15119 1/20 0.42
HSD11B1 P28845 1/20 0.42
GRM2 Q14416 1/20 0.41
HSP90AA1 P07900 1/20 0.41
GABRA1 P14867 1/20 0.41
GABRG2 P18507 1/20 0.41
GABRB3 P28472 1/20 0.41
GABRA5 P31644 1/20 0.41
GABRA3 P34903 1/20 0.41
PDE3B Q13370 1/20 0.41
PDE3A Q14432 1/20 0.41
HSD17B10 Q99714 1/20 0.41
LCK P06239 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17785898 0.85 ERN1 (0.44) ALDH1A1TDP1BRD4ERN1SMARCA2
SCHEMBL26116260 0.85 ERN1 (0.42) ALDH1A1TDP1BRD4ERN1PDK2
SCHEMBL20150143 0.83 ERN1 (0.43) ALDH1A1TDP1BRD4ERN1PDK2
SCHEMBL6372484 0.81 ALDH1A1 (0.50) ALDH1A1TDP1PDK2HSP90AA1PDE3B
SCHEMBL26120840 0.79 ERN1 (0.40) BRD4ERN1SMARCA2SMARCA4ADRA1A
SCHEMBL26118528 0.78 ERN1 (0.39) ALDH1A1BRD4ERN1PDK2LCK
SCHEMBL28712254 0.78 ALDH1A1 (0.54) ALDH1A1TDP1HSP90AA1PDE3BPDE3A
SCHEMBL30490312 0.77 ERN1 (0.38) ALDH1A1BRD4ERN1ADRA1APDK2
SCHEMBL17205693 0.77 SMARCA2 (0.49) BRD4ERN1SMARCA2SMARCA4PDK2
SCHEMBL5913632 0.74 AURKA (0.47) ALDH1A1BRD4ERN1GRM2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6884801-B1 Imidazoline derivatives as alpha-1A adrenoceptor ligands SMITHKLINE BEECHAM CORPORATION (US) 2005-04-26 US disclosed
US-4810282-A 3-ORTHO-(ISOXAZOLYL,ISOTHIAZOLYL, PYRAZOLYL,THIADIAZOLYL, OXADIAZOLYL AND TRIAZOLYL BENZENESULFONUREYLENE-1,2,4-TRIAZOLES E. I. DU PONT DE NEMOURS AND COMPANY (US) 1989-03-07 US disclosed
EP-0083975-B1 HERBICIDAL SULFONAMIDES E.I. DU PONT DE NEMOURS AND COMPANY (US) 1987-11-19 EP disclosed
US-4695311-A Herbicidal sulfonamides E. I. DU PONT DE NEMOURS AND COMPANY (US) 1987-09-22 US disclosed
US-4606755-A Herbicidal sulfonamides E. I. DU PONT DE NEMOURS AND COMPANY (US) 1986-08-19 US disclosed
US-4511392-A N--/PYRIMIDIN-2-YLAMINOCARBENYL/-HETERO-SUBSTITUETED BENZENSESULFO E. I. DU PONT DE NEMOURS AND COMPANY (US) 1985-04-16 US disclosed
EP-0083975-A2 Herbicidal sulfonamides E.I. DU PONT DE NEMOURS AND COMPANY (US) 1983-07-20 EP disclosed