SCHEMBL6375190

SCHEMBL6375190

COc1ncccc1C(O)c1cccs1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.48
MAPT P10636 3/20 0.43
HSD17B10 Q99714 1/20 0.43
CNR2 P34972 1/20 0.42
TOP2A P11388 2/20 0.42
TOP2B Q02880 2/20 0.42
EGFR P00533 1/20 0.42
NPSR1 Q6W5P4 2/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
ALDH1A1 P00352 1/20 0.41
PKM P14618 1/20 0.41
HPGD P15428 1/20 0.41
HTT P42858 1/20 0.41
ATM Q13315 1/20 0.41
CYP3A4 P08684 2/20 0.39
CYP2D6 P10635 2/20 0.39
SLC6A2 P23975 2/20 0.39
SLC6A4 P31645 2/20 0.39
SLC6A3 Q01959 2/20 0.39
PDE4A P27815 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5214224 0.78 TSHR (0.50) TSHRMAPTHSD17B10TOP2ATOP2B
SCHEMBL8198783 0.78 TOP2A (0.54) TSHRMAPTHSD17B10CNR2TOP2A
SCHEMBL23363181 0.75 CYP2D6 (0.45) MAPTALDH1A1HPGDATMCYP3A4
SCHEMBL23363180 0.75 CYP2D6 (0.45) MAPTALDH1A1HPGDATMCYP3A4
SCHEMBL25227231 0.75 CYP2D6 (0.45) MAPTALDH1A1HPGDATMCYP3A4
SCHEMBL29757465 0.75 CYP2D6 (0.45) MAPTALDH1A1HPGDATMCYP3A4
SCHEMBL5381285 0.74 CYP2D6 (0.45) TSHRALDH1A1HPGDATMCYP3A4
SCHEMBL21831822 0.73 SLC6A2 (0.44) MAPTALDH1A1ATMCYP3A4CYP2D6
SCHEMBL26988320 0.73 CYP2D6 (0.44) MAPTALDH1A1HPGDCYP3A4CYP2D6
SCHEMBL30083020 0.71 APLNR (0.44) TSHRHPGDCYP3A4CYP2D6SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1217001-B1 QUINUCLIDINE COMPOUNDS AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT EISAI CO LTD (JP) 2005-12-07 EP disclosed
US-6599917-B1 A squalene-synthesizing enzyme inhibitor, a cholesterol biosynthesis inhibitor and a triglyceride biosynthesis inhibitor EISAI CO., LTD. (JP) 2003-07-29 US disclosed
EP-1217001-A1 QUINUCLIDINE COMPOUNDS AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT Eisai Co., Ltd. (JP) 2002-06-26 EP disclosed