SCHEMBL6380787

SCHEMBL6380787

CCC(C)(C)C(=O)On1c(=O)c2c(ncn2Cc2ccccc2)n(COC(=O)C(C)(C)C)c1=O

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.48
KMT2A Q03164 4/20 0.46
SMN1; SMN2 Q16637 2/20 0.45
ADORA2B P29275 1/20 0.45
RXFP1 Q9HBX9 1/20 0.45
PDE1A P54750 1/20 0.45
PDE1B Q01064 1/20 0.45
PDE1C Q14123 1/20 0.45
POLB P06746 1/20 0.44
HIF1A Q16665 1/20 0.44
MEN1 O00255 2/20 0.44
HPGD P15428 1/20 0.44
TSHR P16473 1/20 0.44
MAPK1 P28482 1/20 0.44
MAPT P10636 1/20 0.42
CNOT7 Q9UIV1 2/20 0.41
USP2 O75604 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2957710 0.86 ALDH1A1 (0.57) ALDH1A1KMT2ASMN1; SMN2ADORA2BRXFP1
SCHEMBL2967449 0.85 PDE1A (0.62) ALDH1A1KMT2ASMN1; SMN2ADORA2BRXFP1
SCHEMBL6383655 0.84 PDE4A (0.35) ALDH1A1KMT2ASMN1; SMN2ADORA2B
SCHEMBL2961214 0.82 POLB (0.64) ALDH1A1KMT2ASMN1; SMN2ADORA2BRXFP1
SCHEMBL5791764 0.82 ALDH1A1 (0.34) ALDH1A1KMT2ASMN1; SMN2MEN1TSHR
SCHEMBL6381761 0.82 SMN1; SMN2 (0.60) ALDH1A1KMT2ASMN1; SMN2ADORA2BRXFP1
SCHEMBL6380785 0.82 KMT2A (0.52) ALDH1A1KMT2ASMN1; SMN2ADORA2BRXFP1
SCHEMBL5718879 0.81 POLB (0.65) ALDH1A1KMT2ASMN1; SMN2ADORA2BRXFP1
SCHEMBL2952786 0.78 BRD4 (0.59) ALDH1A1KMT2APOLBMEN1HPGD
SCHEMBL6379880 0.76 BRD4 (0.54) ALDH1A1KMT2ASMN1; SMN2ADORA2BRXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1557165-A1 COMBINATION DRUG Eisai Co., Ltd. (JP) 2005-07-27 EP disclosed