SCHEMBL6380818

SCHEMBL6380818

CCCCCCCCCCC1C(=O)NC(=O)NC1=O

nearest known ligand 0.60

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.60
KDM4E B2RXH2 1/20 0.60
MEN1 O00255 1/20 0.60
MAPT P10636 1/20 0.60
PKM P14618 1/20 0.60
HPGD P15428 1/20 0.60
KMT2A Q03164 1/20 0.60
LMNA P02545 2/20 0.47
L3MBTL1 Q9Y468 1/20 0.45
HLCS P50747 2/20 0.44
HSD17B10 Q99714 1/20 0.41
CYP1A2 P05177 2/20 0.38
MMP2 P08253 4/20 0.38
MMP9 P14780 4/20 0.38
MMP3 P08254 2/20 0.38
TSHR P16473 1/20 0.37
MMP8 P22894 2/20 0.37
MMP13 P45452 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6381412 1.00 ALDH1A1 (0.60) ALDH1A1KDM4EMEN1MAPTPKM
SCHEMBL472596 1.00 ALDH1A1 (0.60) ALDH1A1KDM4EMEN1MAPTPKM
SCHEMBL21496215 1.00 ALDH1A1 (0.60) ALDH1A1KDM4EMEN1MAPTPKM
SCHEMBL9885892 1.00 ALDH1A1 (0.60) ALDH1A1KDM4EMEN1MAPTPKM
SCHEMBL3911611 0.98 ALDH1A1 (0.62) ALDH1A1KDM4EMEN1MAPTPKM
SCHEMBL572791 0.91 ALDH1A1 (0.64) ALDH1A1KDM4EMEN1MAPTPKM
SCHEMBL472502 0.91 ALDH1A1 (0.70) ALDH1A1KDM4EMEN1MAPTPKM
SCHEMBL1263811 0.89 ALDH1A1 (0.68) ALDH1A1KDM4EMEN1MAPTPKM
Hydrochloric Acid SCHEMBL2722732 0.89 ALDH1A1 (0.62) ALDH1A1KDM4EMEN1MAPTPKM
SCHEMBL1262566 0.89 ALDH1A1 (0.68) ALDH1A1KDM4EMEN1MAPTPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1318406-C New barbituric acid derivatives, processes for their prodn. and pharmaceutical agent contg. same BOEHRINGER MANNHEIM GMBH (DE) 2007-05-30 CN disclosed
CN-1295227-C Barbituric acid derivatives with anti-metastatic and anti-tumor activities ROCH DIAGNOSIS EQUIPMENT AG (DE) 2007-01-17 CN disclosed
EP-0989982-B1 BARBITURIC ACID DERIVATIVES WITH ANTIMETASTATIC AND ANTITUMOR ACTIVITY ROCHE DIAGNOSTICS GMBH (DE) 2005-08-17 EP disclosed
US-6472396-B1 Barbituric acid derivatives, processes for their production and pharmaceutical agents containing these compounds ROCHE DIAGNOSTICS GMBH (DE) 2002-10-29 US disclosed
EP-0869947-B1 BARBITURIC ACID DERIVATIVES, PROCESSES FOR THEIR PRODUCTION AND PHARMACEUTICAL AGENTS CONTAINING THESE COMPOUNDS ROCHE DIAGNOSTICS GMBH (DE) 2002-10-23 EP disclosed
US-6335332-B1 MATRIX METALLOPROTEASE INHIBITORS; CONTRACEPTIVES, ANTIINFLAMMATORY AGENTS ROCHE DIAGNOSTICS GMBH (DE) 2002-01-01 US disclosed
CN-1267296-A Barbituric acid derivatives with anti-metastatic and anti-tumor activities ROCH DIAGNOSIS EQUIPMENT AG (DE) 2000-09-20 CN disclosed
US-6110924-A MATRIX METALLOPROTEASE INHIBITORS ROCHE DIAGNOSTICS GMBH (DE) 2000-08-29 US disclosed
EP-0989982-A1 BARBITURIC ACID DERIVATIVES WITH ANTIMETASTATIC AND ANTITUMOR ACTIVITY Roche Diagnostics GmbH (DE) 2000-04-05 EP disclosed
CN-1209123-A New barbituric acid derivatives, processes for their prodn. and pharmaceutical agent contg. same BOEHRINGER MANNHEIM GMBH (DE) 1999-02-24 CN disclosed
WO-1998058925-A1 BARBITURIC ACID DERIVATIVES WITH ANTIMETASTATIC AND ANTITUMOR ACTIVITY ROCHE DIAGNOSTICS GMBH (DE) 1998-12-30 WO disclosed
EP-0869947-A1 NEW BARBITURIC ACID DERIVATIVES, PROCESSES FOR THEIR PRODUCTION AND PHARMACEUTICAL AGENTS CONTAINING THESE COMPOUNDS Roche Diagnostics GmbH (DE) 1998-10-14 EP disclosed
WO-1997023465-A1 NEW BARBITURIC ACID DERIVATIVES, PROCESSES FOR THEIR PRODUCTION AND PHARMACEUTICAL AGENTS CONTAINING THESE COMPOUNDS BOEHRINGER MANNHEIM GMBH (DE) 1997-07-03 WO disclosed