SCHEMBL6404619

SCHEMBL6404619

Cc1oc(-c2cccc(Cl)c2)nc1CC1(NCC(=O)N2CCCC2C#N)CC1

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.47
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
TP53 P04637 8/20 0.46
MAPT P10636 5/20 0.46
GAA P10253 2/20 0.46
DPP4 P27487 2/20 0.45
HTT P42858 1/20 0.44
PREP P48147 1/20 0.44
USP2 O75604 1/20 0.43
ALOX15 P16050 1/20 0.43
MAPK1 P28482 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL663417 1.00 NPC1 (0.47) NPC1MEN1KMT2ATP53MAPT
SCHEMBL666152 0.90 DPP4 (0.49) DPP4PREP
SCHEMBL4857151 0.88 DPP4 (0.51) DPP4PREP
SCHEMBL665308 0.88 DPP4 (0.51) DPP4PREP
SCHEMBL665317 0.88 DPP4 (0.53) DPP4PREP
SCHEMBL664051 0.88 DPP4 (0.45) DPP4PREP
SCHEMBL664742 0.86 DPP4 (0.46) MEN1KMT2ATP53MAPTDPP4
SCHEMBL6829857 0.86 DPP4 (0.46) MEN1KMT2ATP53MAPTDPP4
SCHEMBL4594320 0.84 DPP4 (0.57) NPC1DPP4
SCHEMBL666221 0.84 DPP4 (0.57) NPC1DPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6861440-B2 DPP IV inhibitors HOFFMANN-LA ROCHE INC. (US) 2005-03-01 US disclosed