SCHEMBL6405875

SCHEMBL6405875

COc1cc(C)ccc1S(=O)(=O)N1CCC(=O)C(C(c2ccccc2)c2ccccc2)C1

nearest known ligand 0.54

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MCOLN3 Q8TDD5 1/20 0.54
TACR1 P25103 12/20 0.49
ALDH1A1 P00352 2/20 0.47
POLB P06746 1/20 0.47
PKM P14618 1/20 0.46
USP2 O75604 2/20 0.45
GAA P10253 1/20 0.45
KMT2A Q03164 1/20 0.45
TSHR P16473 3/20 0.45
MAPK1 P28482 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6412462 0.72 TACR1 (0.55) TACR1
SCHEMBL6412458 0.71 TACR1 (0.53) TACR1
SCHEMBL6408396 0.69 TACR1 (0.53) TACR1
SCHEMBL6408869 0.68 TACR1 (0.85) TACR1
SCHEMBL6408750 0.67 TACR1 (0.84) TACR1
SCHEMBL5069904 0.67 MCOLN3 (0.56) MCOLN3ALDH1A1POLBPKMUSP2
SCHEMBL6407312 0.67 TACR1 (0.70) TACR1
SCHEMBL6410557 0.67 TACR1 (0.68) TACR1
SCHEMBL12719741 0.67 MCOLN3 (0.52) MCOLN3ALDH1A1POLBUSP2KMT2A
SCHEMBL6411916 0.67 TACR1 (0.76) TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050038072-A1 Nitrogeneous cyclic ketone derivative, process for producing the same, and use TAKEDA CHEMICAL INDUSTRIES, LTD. 2005-02-17 US disclosed
EP-1460062-A1 NITROGENOUS CYCLIC KETONE DERIVATIVE, PROCESS FOR PRODUCING THE SAME, AND USE Takeda Chemical Industries, Ltd. (JP) 2004-09-22 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050038072-A1 Nitrogeneous cyclic ketone derivative, process for producing the same, and use BDKRB1, BDKRB2, TACR1 MCOLN3 4643/4885TACR1 3/4885ALDH1A1 1984/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.