SCHEMBL6408380

SCHEMBL6408380

CN1CCC(=O)C(C(c2ccccc2)c2ccc(Cl)cc2)C1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 13/20 0.64
CHRM2 P08172 2/20 0.48
HTR1A P08908 2/20 0.48
ADRA2A P08913 2/20 0.48
CHRM1 P11229 2/20 0.48
DRD1 P21728 2/20 0.48
TBXA2R P21731 2/20 0.48
SLC6A2 P23975 2/20 0.48
SLC6A4 P31645 2/20 0.48
ADRA1A P35348 2/20 0.48
DRD3 P35462 2/20 0.48
SLC6A3 Q01959 2/20 0.48
KCNH2 Q12809 2/20 0.48
BCL2 P10415 1/20 0.48
HRH3 Q9Y5N1 1/20 0.48
CYP2D6 P10635 2/20 0.47
TSHR P16473 1/20 0.47
CYP2C19 P33261 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
SMN1; SMN2 Q16637 3/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6411082 0.94 TACR1 (0.59) TACR1MEN1KMT2A
SCHEMBL6407083 0.91 TACR1 (0.60) TACR1
SCHEMBL6413697 0.80 TACR1 (0.97) TACR1
SCHEMBL6409659 0.80 TACR1 (0.58) TACR1
SCHEMBL6413713 0.78 TACR1 (1.00) TACR1
SCHEMBL6410310 0.77 TACR1 (0.58) TACR1ALDH1A1
SCHEMBL6413686 0.76 TACR1 (0.68) TACR1
SCHEMBL6414888 0.75 TACR1 (0.54) TACR1ALDH1A1CYP3A4HPGD
SCHEMBL6412492 0.72 TACR1 (0.72) TACR1
SCHEMBL4487177 0.71 TACR1 (0.55) TACR1CYP2D6ALDH1A1CYP3A4KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050038072-A1 Nitrogeneous cyclic ketone derivative, process for producing the same, and use TAKEDA CHEMICAL INDUSTRIES, LTD. 2005-02-17 US disclosed
EP-1460062-A1 NITROGENOUS CYCLIC KETONE DERIVATIVE, PROCESS FOR PRODUCING THE SAME, AND USE Takeda Chemical Industries, Ltd. (JP) 2004-09-22 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050038072-A1 Nitrogeneous cyclic ketone derivative, process for producing the same, and use BDKRB1, BDKRB2, TACR1 TACR1 3/4885CHRM2 313/4885HTR1A 172/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.