SCHEMBL6410481

SCHEMBL6410481

CCCc1c(OCCCN2C(=O)NC(C)(c3ccccc3)C2=O)ccc2c(-c3ccccc3)onc12

nearest known ligand 0.60

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 17/20 0.60
NR1H3 Q13133 10/20 0.49
ALDH1A1 P00352 2/20 0.46
GAA P10253 1/20 0.46
TP53 P04637 1/20 0.42
TSHR P16473 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6405303 0.87 NR1H2 (0.65) NR1H2NR1H3ALDH1A1GAA
SCHEMBL6411684 0.86 NR1H2 (0.57) NR1H2NR1H3ALDH1A1GAATP53
SCHEMBL6098553 0.85 NR1H2 (0.62) NR1H2
SCHEMBL6100597 0.82 NR1H2 (0.69) NR1H2NR1H3
SCHEMBL6100301 0.79 NR1H2 (0.61) NR1H2NR1H3ALDH1A1GAA
SCHEMBL6406340 0.79 NR1H2 (0.56) NR1H2NR1H3
SCHEMBL6406547 0.79 NR1H2 (0.59) NR1H2NR1H3
SCHEMBL6407486 0.79 NR1H2 (0.55) NR1H2NR1H3
SCHEMBL1594805 0.77 NR1H2 (0.95) NR1H2NR1H3
SCHEMBL6406183 0.77 NR1H2 (0.42) NR1H2NR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1534696-A1 THERAPEUTIC COMPOUNDS FOR TREATING DYSLIPIDEMIC CONDITIONS Merck & Co., Inc. (US) 2005-06-01 EP claimed
WO-2004011448-A1 THERAPEUTIC COMPOUNDS FOR TREATING DYSLIPIDEMIC CONDITIONS MERCK & CO., INC. (US) 2004-02-05 WO claimed
EP-1534696-A1 THERAPEUTIC COMPOUNDS FOR TREATING DYSLIPIDEMIC CONDITIONS Merck & Co., Inc. (US) 2005-06-01 EP disclosed
WO-2004011448-A1 THERAPEUTIC COMPOUNDS FOR TREATING DYSLIPIDEMIC CONDITIONS MERCK & CO., INC. (US) 2004-02-05 WO disclosed