SCHEMBL6411227

SCHEMBL6411227

COc1ccc(-n2nc(C(C)S(=O)(=O)O)cc2-c2ccccc2)cn1.COc1ccc(-n2nc(CO)cc2-c2ccccc2)cn1

nearest known ligand 0.52

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 7/20 0.52
CA1 P00915 13/20 0.49
CA2 P00918 13/20 0.49
CA9 Q16790 13/20 0.49
PTGS1 P23219 3/20 0.44
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4477596 0.86 PTGS2 (0.57) PTGS2CA1CA2CA9PTGS1
SCHEMBL4476914 0.82 PTGS2 (0.57) PTGS2CA1CA2CA9PTGS1
SCHEMBL4476916 0.79 PTGS2 (0.46) PTGS2CA1CA2CA9PTGS1
SCHEMBL2915550 0.77 PTGS2 (0.57) PTGS2CA1CA2CA9PTGS1
SCHEMBL2941675 0.72 CA1 (0.51) PTGS2CA1CA2CA9PTGS1
SCHEMBL2917637 0.72 MEN1 (0.46) PTGS2CA1CA2CA9PTGS1
SCHEMBL2910437 0.72 RPA1 (0.70) MEN1KMT2A
SCHEMBL5529650 0.70 RPA1 (0.57) CA9MEN1KMT2A
SCHEMBL5147886 0.70 SMO (0.47) MEN1KMT2A
SCHEMBL5149016 0.70 MALT1 (0.45) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1591443-A1 PYRAZOLE DERIVATIVE DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2005-11-02 EP disclosed