SCHEMBL6415733

SCHEMBL6415733

N#Cc1ccccc1C#N.[Li]CCCC

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.50
L3MBTL1 Q9Y468 3/20 0.41
GAA P10253 3/20 0.38
ALDH1A1 P00352 3/20 0.38
HPGD P15428 2/20 0.38
POLB P06746 1/20 0.38
NPC1 O15118 1/20 0.38
CASP3 P42574 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
SENP8 Q96LD8 1/20 0.38
SENP7 Q9BQF6 1/20 0.38
SENP6 Q9GZR1 1/20 0.38
GRM2 Q14416 1/20 0.37
NLRP3 Q96P20 1/20 0.36
KDM4E B2RXH2 2/20 0.35
HTT P42858 1/20 0.35
HSD17B10 Q99714 1/20 0.35
AR P10275 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Octanol SCHEMBL28328490 0.76 ALDH1A1 (0.50) TSHRL3MBTL1GAAALDH1A1HPGD
Alcohol SCHEMBL7573294 0.75 TSHR (0.54) TSHRL3MBTL1GAAALDH1A1HPGD
SCHEMBL2818597 0.74 TSHR (0.63) TSHRGAAALDH1A1HPGDPOLB
Water SCHEMBL27896186 0.74 TSHR (0.63) TSHRGAAALDH1A1HPGDPOLB
SCHEMBL29352197 0.74 TSHR (0.63) TSHRGAAALDH1A1HPGDPOLB
Water SCHEMBL19410621 0.74 TSHR (0.63) TSHRGAAALDH1A1HPGDPOLB
SCHEMBL57480 0.74 TSHR (0.63) TSHRGAAALDH1A1HPGDPOLB
SCHEMBL1726412 0.73 TSHR (0.45) TSHRL3MBTL1ALDH1A1HPGDNPC1
SCHEMBL3568604 0.73 TSHR (0.56) TSHRL3MBTL1GAAALDH1A1HPGD
Naphthalene SCHEMBL11122594 0.73 HTT (0.41) TSHRNPC1RAB9ASMN1; SMN2NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1603918-A1 BORONATED METAL-PHTHALOCYANINES, PROCESS FOR THEIR PREPARATION, PHARMACEUTICAL COMPOSITIONS COMPRISING THEM AND USE THEREOF L. MOLTENI & C. DEI FRATELLI ALITTI SOCIETA' DI ESERCIZIO S.P.A (IT) 2005-12-14 EP disclosed
WO-2004081014-A1 BORONATED METAL-PHTHALOCYANINES, PROCESS FOR THEIR PREPARATION, PHARMACEUTICAL COMPOSITIONS COMPRISING THEM AND USE THEREOF L. MOLTENI & C. DEI FRATELLI ALITTI SOCIETA' DI ESERCIZIO S.P.A. (IT) 2004-09-23 WO disclosed