SCHEMBL6421665

SCHEMBL6421665

CCOC(=O)CC(C=CCCCCc1ccc2c(n1)NCCC2)c1cnc2occc2c1

nearest known ligand 0.54

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ITGAV P06756 20/20 0.54
ITGB3 P05106 12/20 0.54
ITGB6 P18564 9/20 0.44
ITGB8 P26012 7/20 0.44
ITGB5 P18084 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6421661 1.00 ITGAV (0.54) ITGAVITGB3ITGB6ITGB8ITGB5
SCHEMBL6424882 0.87 ITGAV (0.60) ITGAVITGB3ITGB6ITGB8ITGB5
SCHEMBL6424883 0.87 ITGAV (0.60) ITGAVITGB3ITGB6ITGB8ITGB5
SCHEMBL6108062 0.85 ITGAV (0.56) ITGAVITGB3ITGB6ITGB8ITGB5
SCHEMBL6108060 0.85 ITGAV (0.56) ITGAVITGB3ITGB6ITGB8ITGB5
SCHEMBL18105066 0.77 ITGAV (0.60) ITGAVITGB3ITGB6ITGB8ITGB5
SCHEMBL20091226 0.77 ITGAV (0.60) ITGAVITGB3ITGB6ITGB8ITGB5
SCHEMBL6421979 0.76 ITGAV (0.74) ITGAVITGB3ITGB6ITGB8
SCHEMBL6421975 0.76 ITGAV (0.74) ITGAVITGB3ITGB6ITGB8
SCHEMBL6423958 0.76 ITGAV (0.74) ITGAVITGB3ITGB6ITGB8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1040098-B1 INTEGRIN RECEPTOR ANTAGONISTS MERCK & CO INC (US) 2005-04-27 EP disclosed
US-6297249-B1 SUBSTITUTED 2-CARBOXYALKYLPYRIDINES MERCK & CO., INC. 2001-10-02 US disclosed
US-6048861-A OSTEOPOROSIS; BONE DISORDERS; CARDIOVASCULAR DISORDERS; ANTIINFLAMMATROY AGENTS; WOUND HEALING AGENTS MERCK & CO., INC. (US) 2000-04-11 US disclosed