SCHEMBL6422305

SCHEMBL6422305

COc1ccc(S(=O)(=O)C(CCCCc2ccccc2)CC(=O)NO)cc1OCCOCc1ccccc1

nearest known ligand 0.80

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 19/20 0.80
PDE4B Q07343 19/20 0.80
PDE4C Q08493 19/20 0.80
PDE4D Q08499 19/20 0.80
MMP2 P08253 4/20 0.64
MMP3 P08254 4/20 0.64
MMP1 P03956 3/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6422745 0.93 PDE4A (0.89) PDE4APDE4BPDE4CPDE4DMMP2
SCHEMBL6422449 0.92 PDE4A (0.87) PDE4APDE4BPDE4CPDE4DMMP2
SCHEMBL6425155 0.91 PDE4A (0.83) PDE4APDE4BPDE4CPDE4DMMP2
SCHEMBL6822987 0.89 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DMMP2
SCHEMBL6423537 0.88 PDE4A (0.80) PDE4APDE4BPDE4CPDE4DMMP2
SCHEMBL6423418 0.86 PDE4A (0.76) PDE4APDE4BPDE4CPDE4DMMP2
SCHEMBL6423229 0.86 PDE4A (0.76) PDE4APDE4BPDE4CPDE4DMMP2
SCHEMBL6423676 0.85 PDE4A (0.75) PDE4APDE4BPDE4CPDE4DMMP2
SCHEMBL5702974 0.82 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DMMP2
SCHEMBL6424717 0.82 PDE4A (0.69) PDE4APDE4BPDE4CPDE4DMMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0960096-B1 SUBSTITUTED BETA-THIOCARBOXYLIC ACIDS AVENTIS PHARMA INC (US) 2005-04-06 EP claimed
US-6306873-B1 Substituted β-thiocarboxylic acids AVENTIS PHARMACEUTICALS PRODUCTS INC. 2001-10-23 US claimed
EP-0960096-A1 SUBSTITUTED $g(b)-THIOCARBOXYLIC ACIDS RHONE-POULENC RORER PHARMACEUTICALS, INC. (US) 1999-12-01 EP claimed
WO-1998032734-A1 SUBSTITUTED β-THIOCARBOXYLIC ACIDS RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1998-07-30 WO claimed
EP-0960096-B1 SUBSTITUTED BETA-THIOCARBOXYLIC ACIDS AVENTIS PHARMA INC (US) 2005-04-06 EP disclosed
EP-1486486-A2 Substituted B-thiocarboxylic acids Aventis Pharmaceuticals Inc. (US) 2004-12-15 EP disclosed
US-6306873-B1 Substituted β-thiocarboxylic acids AVENTIS PHARMACEUTICALS PRODUCTS INC. 2001-10-23 US disclosed
EP-0960096-A1 SUBSTITUTED $g(b)-THIOCARBOXYLIC ACIDS RHONE-POULENC RORER PHARMACEUTICALS, INC. (US) 1999-12-01 EP disclosed
WO-1998032734-A1 SUBSTITUTED β-THIOCARBOXYLIC ACIDS RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1998-07-30 WO disclosed