SCHEMBL6427644

SCHEMBL6427644

CC(C(=O)O)c1ccc(C#Cc2ccc3c(c2)C(C)(C)CCC3O)cc1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
RARB P10826 10/20 0.47
RARG P13631 10/20 0.47
RARA P10276 8/20 0.47
CYP26A1 O43174 1/20 0.47
CYP3A4 P08684 1/20 0.47
CRABP2 P29373 1/20 0.47
PTGS1 P23219 7/20 0.36
PTGS2 P35354 7/20 0.36
RXRA P19793 1/20 0.36
RXRB P28702 1/20 0.36
MT-CO1 P00395 1/20 0.36
MT-CO2 P00403 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4517591 0.85 RARB (0.41) RARBRARGRARACYP26A1CYP3A4
SCHEMBL5737254 0.84 RARB (0.67) RARBRARGRARACYP26A1CYP3A4
SCHEMBL4517593 0.83 RARB (0.39) RARBRARGRARACYP26A1CYP3A4
SCHEMBL6426334 0.81 RARA (0.38) RARBRARGRARACYP26A1CYP3A4
SCHEMBL5736773 0.81 CYP26A1 (0.47) RARBRARGRARACYP26A1CYP3A4
SCHEMBL6426143 0.78 RARB (0.46) RARBRARGRARACYP26A1CYP3A4
SCHEMBL4508295 0.77 RARB (0.38) RARBRARGRARACYP26A1CYP3A4
SCHEMBL7640501 0.76 RARB (0.52) RARBRARGRARACYP26A1CYP3A4
SCHEMBL4521595 0.76 RARB (0.36) RARBRARGRARACYP26A1CYP3A4
SCHEMBL4521601 0.75 RARB (0.35) RARBRARGRARACYP26A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6855512-B2 Methods for identifying inhibitors of cytochrome P450RAI ALLERGAN, INC. (US) 2005-02-15 US disclosed
US-6369261-B1 CYCLOPROPYLBENZENE DERIVATIVE OF ACIDS OR ESTERS ALLERGAN SALES, INC. 2002-04-09 US disclosed
US-6369225-B1 ENZYME INHIBITORS ALLERGAN SALES, INC. 2002-04-09 US disclosed
US-6303785-B1 SUBSTITUTED N-CYCLOPROPYLTETRAHYDROISOQUINOLINES ALLERGAN SALES, INC. 2001-10-16 US disclosed