SCHEMBL6428

SCHEMBL6428

O=[N+]([O-])c1ccccc1NC[C@@H]1CCNC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KAT2B Q92831 2/20 0.46
MAPK1 P28482 4/20 0.44
L3MBTL1 Q9Y468 3/20 0.44
TDP1 Q9NUW8 2/20 0.44
ALDH1A1 P00352 1/20 0.44
CASP7 P55210 1/20 0.44
MAPT P10636 4/20 0.44
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
PRKCQ Q04759 1/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
KDM1A O60341 1/20 0.42
MAOB P27338 1/20 0.42
SLC6A2 P23975 1/20 0.42
SLC6A4 P31645 1/20 0.42
IDO1 P14902 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13319008 1.00 KAT2B (0.46) KAT2BMAPK1L3MBTL1TDP1ALDH1A1
Hydrochloric Acid SCHEMBL11909173 0.99 KAT2B (0.47) KAT2BMAPK1L3MBTL1TDP1ALDH1A1
SCHEMBL13834721 0.82 MEN1 (0.50) ALDH1A1MAPTCYP3A4CYP2C9PRKCQ
SCHEMBL13319009 0.81 KAT2B (0.51) KAT2BMAPK1L3MBTL1TDP1ALDH1A1
Hydrochloric Acid SCHEMBL13834520 0.81 MEN1 (0.49) ALDH1A1MAPTCYP3A4CYP2C9PRKCQ
Hydrochloric Acid SCHEMBL6379 0.81 BRD3 (0.43) TDP1ALDH1A1MAPTCYP3A4CYP2C9
Hydrochloric Acid SCHEMBL6092 0.81 CHRM3 (0.41) MAPK1ALDH1A1MAPTPRKCQSMN1; SMN2
SCHEMBL23997424 0.80 ALDH1A1 (0.51) KAT2BMAPK1L3MBTL1TDP1ALDH1A1
SCHEMBL13834543 0.80 NPC1 (0.49) MAPTCYP3A4CYP2C9PRKCQNPC1
SCHEMBL2010060 0.80 RPS6KB1 (0.41) L3MBTL1ALDH1A1CYP3A4CYP2C9PRKCQ

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2493310-A1 BENZIMIDAZOLES AS FATTY ACID SYNTHASE INHIBITORS GlaxoSmithKline LLC (US) 2012-09-05 EP disclosed
WO-2011056635-A1 BENZIMIDAZOLES AS FATTY ACID SYNTHASE INHIBITORS GLAXOSMITHKLINE LLC (US) 2011-05-12 WO disclosed