SCHEMBL6428993

SCHEMBL6428993

Cc1c(N)cccc1-n1ccnn1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 13/20 0.44
CYP3A4 P08684 1/20 0.43
TSHR P16473 1/20 0.43
PIK3CA P42336 1/20 0.43
KEAP1 Q14145 1/20 0.40
ALDH1A1 P00352 1/20 0.37
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
CHRNB2 P17787 1/20 0.36
CYP2B6 P20813 1/20 0.36
MAOA P21397 1/20 0.36
CYP2C19 P33261 1/20 0.36
CHRNA4 P43681 1/20 0.36
HTR3A P46098 1/20 0.36
EGLN2 Q96KS0 1/20 0.35
KDM4E B2RXH2 1/20 0.35
MEN1 O00255 1/20 0.35
USP2 O75604 1/20 0.35
TP53 P04637 1/20 0.35
GAA P10253 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27984977 0.82 NOTUM (0.43) NOTUMKEAP1CYP1A2CYP2C9CHRNB2
SCHEMBL18378736 0.82 NOTUM (0.47) NOTUMTSHRKEAP1ALDH1A1CYP1A2
SCHEMBL454021 0.82 GAA (0.47) NOTUMKEAP1CYP1A2CYP2C9CHRNB2
SCHEMBL3387244 0.79 NOTUM (0.53) NOTUMTSHRKEAP1ALDH1A1CYP1A2
SCHEMBL27613715 0.79 NOTUM (0.44) NOTUMKEAP1ALDH1A1CYP1A2CYP2C9
SCHEMBL22702085 0.79 NOTUM (0.47) NOTUMKEAP1CYP1A2CYP2C9CHRNB2
SCHEMBL15774805 0.79 NOTUM (0.45) NOTUMKEAP1CYP1A2CYP2C9CHRNB2
SCHEMBL7111602 0.79 NOTUM (0.44) NOTUMKEAP1CYP1A2CYP2C9CHRNB2
SCHEMBL21376045 0.79 NOTUM (0.49) NOTUMKEAP1CYP1A2CYP2C9CHRNB2
SCHEMBL17194959 0.77 MAPK1 (0.50) NOTUMCYP3A4TSHRPIK3CAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050288347-A1 Certain triazole-based compounds, compositions, and uses thereof AGRIUS GROUP, LLC. 2005-12-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050288347-A1 Certain triazole-based compounds, compositions, and uses thereof ABCG2, ATP5ME, DNTT NOTUM 607/4885CYP3A4 25/4885TSHR 3470/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.