SCHEMBL6429299

SCHEMBL6429299

Cc1cccc2c(C(=O)O)cc(-c3ccccc3)nc12

nearest known ligand 0.80

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.80
LMNA P02545 2/20 0.80
HTT P42858 1/20 0.80
PDE10A Q9Y233 2/20 0.69
PPARA Q07869 1/20 0.65
PLAUR Q03405 1/20 0.65
POLB P06746 1/20 0.64
SMN1; SMN2 Q16637 1/20 0.63
TP53 P04637 1/20 0.60
MAPT P10636 1/20 0.60
DHODH Q02127 1/20 0.60
ALDH1A1 P00352 1/20 0.59
HSD17B10 Q99714 1/20 0.59
CCR6 P51684 1/20 0.56
NPC1 O15118 1/20 0.56
AURKA O14965 1/20 0.55
PTGER4 P35408 1/20 0.55
AKR1C3 P42330 1/20 0.55
AKR1C2 P52895 1/20 0.55
AKR1C1 Q04828 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Benzaldehyde SCHEMBL22471883 0.91 KDM4E (0.68) KDM4ELMNAHTTPDE10APPARA
SCHEMBL31620698 0.89 KDM4E (1.00) KDM4ELMNAHTTPDE10APPARA
SCHEMBL11810641 0.86 PDE10A (0.70) KDM4ELMNAHTTPDE10APPARA
SCHEMBL8324266 0.86 KDM4E (0.64) KDM4ELMNAHTTPDE10APPARA
SCHEMBL13958056 0.84 CCR6 (0.68) KDM4ELMNAHTTPDE10APPARA
SCHEMBL8619739 0.82 PPARA (0.69) KDM4ELMNAHTTPDE10APPARA
SCHEMBL28019600 0.82 CCR6 (0.67) KDM4ELMNAHTTPDE10APPARA
SCHEMBL22471898 0.82 AURKA (0.78) KDM4ELMNAHTTPDE10APPARA
SCHEMBL8619775 0.82 PPARA (0.64) KDM4ELMNAHTTPDE10APPARA
SCHEMBL10758255 0.82 PDE10A (0.64) KDM4ELMNAHTTPDE10APPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4617270-A1 ISOINDOLINONE DERIVATIVE HAVING QUINOLINE AMIDE STRUCTURE, AND USE THEREOF Oncord Bio Inc (KR) 2025-09-17 EP disclosed
CN-120152966-A Isoindolinone derivative with quinolinamide structure and application thereof 昂科德生物株式会社 2025-06-13 CN disclosed
WO-2024101764-A1 ISOINDOLINONE DERIVATIVE HAVING QUINOLINE AMIDE STRUCTURE, AND USE THEREOF 주식회사 온코드바이오 2024-05-16 WO disclosed
US-20220169640-A1 PRODUCTION METHOD OF QUINOLINECARBOXAMIDE DERIVATIVE OR PRODUCTION INTERMEDIATE THEREOF KABUSHIKI KAISHA YAKULT HONSHA (JP) 2022-06-02 US disclosed
EP-3943159-A1 PRODUCTION METHOD OF QUINOLINECARBOXAMIDE DERIVATIVE OR PRODUCTION INTERMEDIATE THEREOF Kabushiki Kaisha Yakult Honsha (JP) 2022-01-26 EP disclosed
WO-2005118580-A2 TRICYCLIC COMPOUNDS AS INHIBITORS OF THE HYPOXIC SIGNALING PATHWAY THE GOVERNMENT OF THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH (US) 2005-12-15 WO disclosed
US-6906193-B2 N-type calcium channel antagonists for the treatment of pain ASTRAZENECA AB (SE) 2005-06-14 US disclosed
US-20040053964-A1 N-type calcium channel antagonists for the treatment of pain ASTRAZENECA AB (SE) 2004-03-18 US disclosed
EP-1339689-A1 N-TYPE CALCIUM CHANNEL ANTAGONISTS FOR THE TREATMENT OF PAIN AstraZeneca AB (SE) 2003-09-03 EP disclosed
WO-2002036568-A1 N-TYPE CALCIUM CHANNEL ANTAGONISTS FOR THE TREATMENT OF PAIN ASTRAZENECA AB (SE) 2002-05-10 WO disclosed
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed
EP-0206802-B1 SUBSTITUTED QUINOLINE DERIVATIVES CANCER RESEARCH CAMPAIGN TECHNOLOGY LIMITED (GB) 1993-09-01 EP disclosed
US-4904659-A Substituted quinoline derivatives and pharmaceutical compositions thereof DEVELOPMENT FINANCE CORPORATION OF NEW ZELAND (NZ) 1990-02-27 US disclosed
EP-0206802-A2 Substituted quinoline derivatives CANCER RESEARCH CAMPAIGN TECHNOLOGY LIMITED (GB) 1986-12-30 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220169640-A1 PRODUCTION METHOD OF QUINOLINECARBOXAMIDE DERIVATIVE OR PRODUCTION INTERMEDIATE THEREOF BCKDK, CBR3, NQO2 KDM4E 363/4885LMNA 1893/4885HTT 2685/4885
US-20040053964-A1 N-type calcium channel antagonists for the treatment of pain CACNA1E, CACNA1B, CACNA1A KDM4E 4425/4885LMNA 3096/4885HTT 2827/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.