SCHEMBL6429617

SCHEMBL6429617

CCO/C=C(\C(N)=O)c1ccc(Br)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OGG1 O15527 1/20 0.41
MAOB P27338 1/20 0.40
MAPT P10636 4/20 0.40
KMT2A Q03164 3/20 0.40
LMNA P02545 3/20 0.40
NPSR1 Q6W5P4 3/20 0.40
MEN1 O00255 2/20 0.40
MAPK1 P28482 2/20 0.40
S1PR4 O95977 1/20 0.40
S1PR1 P21453 1/20 0.40
HPGD P15428 2/20 0.39
RAB9A P51151 2/20 0.39
NPC1 O15118 1/20 0.39
CES2 O00748 1/20 0.38
CES1 P23141 1/20 0.38
HTT P42858 2/20 0.38
GSK3B P49841 2/20 0.38
POLB P06746 2/20 0.38
ALDH1A1 P00352 3/20 0.38
PARP10 Q53GL7 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL94197 0.83 ALDH1A1 (0.42) MAPTKMT2ALMNANPSR1MEN1
SCHEMBL94199 0.83 ALDH1A1 (0.42) MAPTKMT2ALMNANPSR1MEN1
SCHEMBL11261744 0.73 KMT2A (0.39) OGG1MAOBMAPTKMT2ALMNA
SCHEMBL11092095 0.73 KMT2A (0.39) OGG1MAOBMAPTKMT2ALMNA
SCHEMBL11092100 0.73 KMT2A (0.39) OGG1MAOBMAPTKMT2ALMNA
SCHEMBL27792518 0.70 KMT2A (0.57) MAOBMAPTKMT2ALMNANPSR1
SCHEMBL24788880 0.70 KMT2A (0.46) MAOBMAPTKMT2ALMNANPSR1
SCHEMBL30747063 0.69 AKR1C1 (0.48) MAPTKMT2ALMNAMEN1MAPK1
SCHEMBL18812994 0.69 AKR1C1 (0.48) MAPTKMT2ALMNAMEN1MAPK1
SCHEMBL2384544 0.69 KMT2A (0.55) MAOBMAPTKMT2ALMNANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1558578-A1 NOVEL ALKYNE COMPOUNDS HAVING AN MCH ANTAGONISTIC EFFECT AND MEDICAMENTS CONTAINING THESE COMPOUNDS BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2005-08-03 EP disclosed
WO-2004039780-A1 NOVEL ALKYNE COMPOUNDS HAVING AN MCH ANTAGONISTIC EFFECT AND MEDICAMENTS CONTAINING THESE COMPOUNDS BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2004-05-13 WO disclosed